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Cytokine receptors

StructureProduct infoAvailabilityQuantity / Price
BRC1245
Product IDBRC1245
Product classBioreference compound
CAS number98-79-3
MW129.1
Synonyms
NSC 143034; Oxoproline; Glutiminic acid; Pidolidone; Pidolic Acid;
Transport conditionsNormal

L-Pyroglutamic acid

L-Pyroglutamic acid is an amino acid that is used in the synthesis of peptides. It is cyclooxygenase inhibitor.

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BRC1066
Product IDBRC1066
Product classBioreference compound
CAS number498-02-2
MW166.2
Synonyms
NSC 209524; NSC 2146;
Transport conditionsNormal

Apocynin

Apocynin is a methoxy-substituted catechol that is commonly used as a selective NADPH-oxidase inhibitor with IC50 of 10 μM. Acts as an antioxidant in endothelial cells and vascular smooth muscle cells.

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BRC0133
Product IDBRC0133
Product classBioreference compound
CAS number51-43-4
MW183.2
Synonyms
Adrenalin; L-epinephrine; Levoepinephrine;
Transport conditionsNormal

Epinephrine

Epinephrine is indicated for intravenous injection in treatment of acute hypersensitivity, treatment of acute asthmatic attacks to relieve bronchospasm, and treatment and prophylaxis of cardiac arrest and attacks of transitory atrioventricular heart block with syncopal seizures (Stokes-Adams Syndrome).

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BRC1319
Product IDBRC1319
Product classBioreference compound
CAS number515-13-9
MW204.4
Synonyms
Levo-β-elemene;
Transport conditionsNormal

β-Elemen

β-Elemene is a natural sesquiterpene, inhibits the proliferation of a wide range of tumors. It has antioxidant and antimicrobial properties.

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BRC0999
Product IDBRC0999
Product classBioreference compound
CAS number66-84-2
MW215.6
Synonyms
Chitosamine;
Transport conditionsNormal

Glucosamine Hydrochloride

Glucosamine is an amino sugar and a prominent precursor in the biochemical synthesis of glycosylated proteins and lipids.

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BRC1320
Product IDBRC1320
Product classBioreference compound
CAS number2482-00-0
MW228.3
Synonyms
NIH 11035; NSC 56332;
Transport conditionsNormal

Agmatine sulfate

Agmantine is a natural metabolite of the arginine. It binds to human adrenergic receptors and imidazoline (I) receptors. Agmatine acts as an antagonist of the NMDA receptor and nicotinic acetylcholine receptors. It is an antagonist of the serotonin receptor subtype 5-HT3 and blocks ATP-sensitive potassium channels. Agmatine competitively inhibits neuronal, macrophage, endothelial, and inducible nitric oxide synthase and irreversibly inactivates neuronal NOS in the presence of calmodulin.

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BRC0718
Product IDBRC0718
Product classBioreference compound
CAS number22071-15-4
MW254.3
Synonyms
Orudis; Oruvail;
Transport conditionsNormal

Ketoprofen

Ketoprofen is a nonsteroidal anti-inflammatory agent with analgesic and antipyretic properties. It is used to treat rheumatoid arthritis, osteoarthritis, dysmenorrhea, and alleviate moderate pain. Ketoprofen is a non-selective NSAID exhibiting IC50 values of 0.5 µM and 2.33 µM for human recombinant COX-1 and COX-2, respectively.

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BRC0121
Product IDBRC0121
Product classBioreference compound
CAS number50-35-1
MW258.2
Synonyms
Thalomid, Distaval, Softenon, Talimol,
Transport conditionsNormal
Restrictions Included in California Proposition 65 list  WARNING! This product contains a chemical known to the State of California to cause birth defects or other reproductive harm. For more information go to www.P65Warnings.ca.gov.

Thalidomide

Thalidomide is an immunomodulatory agent with a spectrum of activity that is not fully characterized. Thalidomide is racemic — it contains both left and right handed isomers in equal amounts: one enantiomer is effective against morning sickness, and the other is teratogenic.

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BRC0780
Product IDBRC0780
Product classBioreference compound
CAS number191732-72-6
MW259.3
Synonyms
CC-5013, CDC 501, IMid-1, IMiD3, ENMD 0997
Transport conditionsNormal

Lenalidomide

Lenalidomide is a thalidomide analogue. It is immunomodulatory agent possessing antiangiogenic properties.

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BRC1295
Product IDBRC1295
Product classBioreference compound
CAS number51298-62-5
MW269.7
Synonyms
Transport conditionsNormal

L-NAME hydrochloride

L-NAME hydrochloride is a nonselective inhibitor of nitric oxide synthetases.

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BRC0759
Product IDBRC0759
Product classBioreference compound
CAS number1110650-72-0
MW354.4
Synonyms
Transport conditionsNormal

HFI-419

HFI-419 is a substrate competitive inhibitor of insulin-regulated aminopeptidase (IRAP) activity (Ki = 0.48 µM against 25 µM Leu-AMC).

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BRC0699
Product IDBRC0699
Product classBioreference compound
CAS number903591-53-7
MW413.7
Synonyms
Transport conditionsNormal

N-[5-[2-Chloro-5-(trifluoromethyl)phenyl]-2-pyrazinyl]-2,6-difluorobenzamide

The compound is cytokine and calcium channel inhibitor (IC50 = 2 nM).

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BRC0293
Product IDBRC0293
Product classBioreference compound
CAS number155148-31-5
MW502.8
Synonyms
AMD3100, LM3100, Mozobil,
Transport conditionsNormal

Plerixafor

Plerixafor is a hematopoietic stem cell mobilizer. It is used to stimulate the release of stem cells from the bone marrow into the blood in patients with non-Hodgkin lymphoma and multiple myeloma for the purpose of stimulating the immune system. Plerixafor inhibits the CXCR4 chemokine receptors on CD34+ cells and reversibly blocks binding of the ligand, stromal cell-derived factor-1-alpha (SDF-1α).

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BRC0026
Product IDBRC0026
Product classBioreference compound
CAS number376348-65-1
MW513.7
Synonyms
Selzentry, Celsentri, UK 427857
Transport conditionsNormal

Maraviroc

Maraviroc is a chemokine receptor antagonist drug developed by the drug company Pfizer that is designed to act against HIV by interfering with the interaction between HIV and CCR5. Maraviroc is an entry inhibitor and works by blocking HIV from entering human cells. Specifically maraviroc is a selective, slowly reversible, small molecule antagonist of the interaction between human CCR5 and HIV-1 gp120.

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BRC0003
Product IDBRC0003
Product classBioreference compound
CAS number50-63-5
MW515.9
Synonyms
Aralen, Artrichin, Bemaphate, Capquin, Malarex, Nivaquine B, Resoquine, Reumachlor, Sanoquin
Transport conditionsNormal

Chloroquine diphosphate

Chloroquine is the prototype anti malarial drug, most widely used to treat all types of malaria except for disease caused by chloroquine resistant Plasmodium falciparum. Chloroquine inhibits the parasitic enzyme heme polymerase that converts the toxic heme into non-toxic hemazoin, thereby resulting in the accumulation of toxic heme within the parasite. It may also interfere with the biosynthesis of nucleic acids.

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BRC0581
Product IDBRC0581
Product classBioreference compound
CAS number129453-61-8
MW606.8
Synonyms
ICI 182780, ZD 182780, ZD 9238
Transport conditionsNormal

Fulvestrant

Fulvestrant is an estrogen receptor antagonist (IC50 = 0.29 nM) with no agonist effects, which works both by down-regulating and by degrading the estrogen receptor.

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