EnamineStore

Welcome, Guest
Tutorials

Angiotensin receptor

StructureProduct infoAvailabilityQuantity / Price
BRC0890
Product IDBRC0890
Product classBioreference compound
CAS number62571-86-2
MW217.3
Synonyms
C09AA01, SA-333, SQ-14225
Transport conditionsNormal
Restrictions Included in California Proposition 65 list  WARNING! This product contains a chemical known to the State of California to cause health damage. For more information go to www.P65Warnings.ca.gov.

Captopril

Captopril is a potent, competitive inhibitor of angiotensin-converting enzyme (ACE), the enzyme responsible for the conversion of angiotensin I (ATI) to angiotensin II (ATII). ATII regulates blood pressure and is a key component of the renin-angiotensin-aldosterone system (RAAS).

Product Page

In Stock(5 business days)  
BRC0632
Product IDBRC0632
Product classBioreference compound
CAS number23113-43-1
MW267.5
Synonyms
NSC 68982, Wy 8678
Transport conditionsNormal

Guanabenz hydrochloride

Guanabenz is a centrally acting α-2 adrenergic agonist and IGRS (imidazoline I2 binding site) selective ligand, indicated for treatment of hypertension.

Product Page

In Stock(5 business days)  
BRC0509
Product IDBRC0509
Product classBioreference compound
CAS number82158-86-9
MW319.4
Synonyms
Kinedak; ONO 2235; Sorbista;
Transport conditionsNormal

Epalrestat

Epalrestat is a carboxylic acid-based inhibitor of aldose reductase (IC50 = 0.01-15 μM). Epalrestat has been shown to reduce oxidative stress in type 2 diabetic patients, significantly decreasing lipid hydroperoxide levels in erythrocytes when administered at 150 mg/day.

Product Page

In Stock(5 business days)  
BRC0095
Product IDBRC0095
Product classBioreference compound
CAS number84680-54-6
MW384.4
Synonyms
Enalapril acid, MK-422 Dihydrate
Transport conditionsNormal

Enalaprilat dihydrate

Enalaprilat is the active metabolite of the orally available pro-drug, enalapril. Used in the treatment of hypertension, enalapril is an ACE inhibitor that prevents Angiotensin Converting Enzyme (ACE) from transforming angiotensin I into angiotensin II.

Product Page

In Stock(5 business days)  
BRC0855
Product IDBRC0855
Product classBioreference compound
CAS number76547-98-3
MW405.5
Synonyms
MK 521, MK 522
Transport conditionsNormal
Restrictions Included in California Proposition 65 list  WARNING! This product contains a chemical known to the State of California to cause health damage. For more information go to www.P65Warnings.ca.gov.

Lisinopril

Lisinopril is a potent, competitive inhibitor of angiotensin-converting enzyme, the enzyme responsible for the conversion of angiotensin I (ATI) to angiotensin II (ATII). ATII is a key component of the renin-angiotensin-aldosterone system (RAAS).

Product Page

In Stock(5 business days)  
BRC0716
Product IDBRC0716
Product classBioreference compound
CAS number87333-19-5
MW416.5
Synonyms
Corpril, Delix, Ecator, HOE 498
Transport conditionsNormal
Restrictions Included in California Proposition 65 list  WARNING! This product contains a chemical known to the State of California to cause health damage. For more information go to www.P65Warnings.ca.gov.

Ramipril

Ramipril is non-peptide, competitive angiotensin converting enzyme (ACE) inhibitor (IC50 = 5 nM). It is prodrug which is hydrolyzed in vivo to the active metabolite ramiprilat. Displays protective effects on endothelium against high-glucose induced dysfunction.

Product Page

In Stock(5 business days)  
BRC0416
Product IDBRC0416
Product classBioreference compound
CAS number114798-26-4
MW422.9
Synonyms
Lortaan, DuP-753, MK 954
Transport conditionsNormal

Losartan

Losartan is the first of a class of antihypertensive agents called angiotensin II receptor blockers (ARBs). Losartan and its longer acting active metabolite, E-3174, are specific and selective type-1 angiotensin II receptor (AT1) antagonists which block the blood pressure increasing effects angiotensin II via the renin-angiotensin-aldosterone system (RAAS).

Product Page

In Stock(5 business days)  
BRC0028
Product IDBRC0028
Product classBioreference compound
CAS number144689-24-7
MW446.5
Synonyms
Erastapex, Golme, Olmetec, WinBP
Transport conditionsNormal

Olmesartan

Olmesartan is a specific angiotensin II type 1 (AT1) receptor antagonist, which blocks the blood pressure increasing effects of angiotensin II via the renin-angiotensin-aldosterone system (RAAS).

Product Page

In Stock(5 business days)  
BRC0850
Product IDBRC0850
Product classBioreference compound
CAS number82586-55-8
MW475.0
Synonyms
C09AA06
Transport conditionsNormal

Quinapril hydrochloride

Quinapril hydrochloride is a prodrug, angiotensin-converting enzyme (ACE) inhibitor. It is metabolized to quinaprilat (quinapril diacid) following oral administration. Quinaprilat is a competitive inhibitor of ACE, the enzyme responsible for the conversion of angiotensin I (ATI) to angiotensin II (ATII).

Product Page

In Stock(5 business days)  
BRC0679
Product IDBRC0679
Product classBioreference compound
CAS number144701-48-4
MW514.6
Synonyms
BIBR 277, BIBR 277SE, Kinzalmono, Micardis, Pritor, Telday
Transport conditionsNormal

Telmisartan

Telmisartan is a non-peptide AT1 angiotensin receptor antagonist (Ki = 3.7 nM). Exhibits antihypertensive activity in a renin-dependent model of hypertension. Telmisartan also have PPAR-gamma agonistic properties (EC50 = 4 nM) that could potentially confer beneficial metabolic effects.

Product Page

In Stock(5 business days)  
BRC0093
Product IDBRC0093
Product classBioreference compound
CAS number144689-63-4
MW558.6
Synonyms
Benicar, Cs 866,
Transport conditionsNormal

Olmesartan medoxomil

Prodrug metabolised in vivo to Olmesartan, a selective non-peptide angiotensin II type I receptor (AT1) antagonist. Selectively inhibits angiotensin II binding to AT1 receptors in bovine adrenal cortical membranes (IC50 = 7.7 nM), with no effect on AT2 receptors.

Product Page

In Stock(5 business days)  
BRC0681
Product IDBRC0681
Product classBioreference compound
CAS number98048-97-6
MW563.7
Synonyms
Fozitec
Transport conditionsNormal

Fosinopril

Fosinopril is an inhibitor of Angiotensin-converting enzyme (ACE). In nature, ACE converts angiotensin I to angiotensin II, which causes blood vessels to constrict, and thereby increasing blood pressure.

Product Page

In Stock(5 business days)  
BRC0334
Product IDBRC0334
Product classBioreference compound
CAS number145040-37-5
MW610.7
Synonyms
TCV-116
Transport conditionsNormal

Candesartan Cilexetil

Candesartan cilexetil is a prodrug of the potent, long-acting, and selective angiotensin II type 1 receptor (AT1) antagonist, candesartan.

Product Page

In Stock(5 business days)  
Display records per page

 

x
x