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GABA receptors

StructureProduct infoAvailabilityQuantity / Price
BRC0254
Product IDBRC0254
Product classBioreference compound
CAS number142-63-2
MW86.1
Synonyms
Diethylenediamine, Piperazidine, Piperazin, Antepar, Uvilon, Vermidol, Vermizine
Transport conditionsNormal

Piperazine Hexahydrate

Piperazine is a GABA receptor agonist.

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BRC0928
Product IDBRC0928
Product classBioreference compound
CAS number68506-86-5
MW129.2
Synonyms
CPP-109; MDL 71,754; MDL-71754; RMI-71754; GVG; Sabril™; γ-Vinyl GABA;
Transport conditionsNormal

Vigabatrin

Vigabatrin is a structural analogue of gamma-aminobutyric acid, irreversible inhibitor of 4-aminobutyrate transaminase, the enzyme responsible for the catabolism of gamma-aminobutyric acid.

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BRC1062
Product IDBRC1062
Product classBioreference compound
CAS number4393-06-0
MW134.2
Synonyms
Phenylvinylcarbinol; α-Phenylallyl alcohol; α-Vinylbenzyl alcohol;
Transport conditionsNormal

NSC 167595

NSC 167595 is an anti-allergic agent.

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BRC1417
Product IDBRC1417
Product classBioreference compound
CAS number3687-18-1
MW139.2
Synonyms
Alzhemed; Homotaurine; NC 758; NSC 77071; γ-Aminopropylsulfonic acid;
Transport conditionsNormal

Tramiprosate

Tramiprosate is a GABA mimetic that targets soluble amyloid β (Aβ) and maintains Aβ in a non-fibrillar form. Decreases Aβ42-induced neuronal death and inhibit amyloid deposition in vitro. Decreases brain amyloid plaque load by 30%, increases tau polymerization and is brain penetrant. Also, a GABA analog that protects against the convulsant and cytotoxic activity of kainic acid in vivo.

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BRC1029
Product IDBRC1029
Product classBioreference compound
CAS number59-50-7
MW142.6
Synonyms
NSC 4166; Neopredisan; Parol; Raschit; PCMC;
Transport conditionsNormal

Chlorocresol

Chlorocresol is a chlorinated phenol which is used as an antiseptic and preservative.

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BRC1033
Product IDBRC1033
Product classBioreference compound
CAS number64-65-3
MW155.2
Synonyms
Mikedimide; NP 13; NSC 168667; NSC 58187; Zentraleptin;
Transport conditionsNormal

Bemegride

Bemegride is a central nervous system stimulant and antidote for barbiturate poisoning as its chemoreceptor agonism increases mean tidal volume, thereby increasing respiration and the concentration of O2 in blood.

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BRC0909
Product IDBRC0909
Product classBioreference compound
CAS number182485-36-5
MW161.1
Synonyms
Transport conditionsNormal

TPMPA

TPMPA is GABA receptor antagonist.

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BRC0692
Product IDBRC0692
Product classBioreference compound
CAS number76-38-0
MW165.0
Synonyms
DA-759; NSC-110432;
Transport conditionsNormal

Methoxyflurane

Methoxyflurane is an anesthetic used for induction and maintenance of general anesthesia. It induces muscle relaxation and reduces pains sensitivity by altering tissue excitability.

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BRC0615
Product IDBRC0615
Product classBioreference compound
CAS number2078-54-8
MW178.3
Synonyms
ICI 35868; Disoprivan; Disoprofol;
Transport conditionsNormal

Propofol

Propofol is a sedative-hypnotic agent for use in the induction and maintenance of anesthesia or sedation. It acts as a potentiator of the GABAA receptor.

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BRC0958
Product IDBRC0958
Product classBioreference compound
CAS number79416-27-6
MW181.6
Synonyms
Metvixia; Visonac; MAL;
Transport conditionsNormal

Methyl aminolevulinate Hydrochloride

Methyl aminolevulinate hydrochloride is a prodrug that is metabolized to Protoporphyrin IX (a photosensitizer) used in photodynamic therapy.

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BRC0823
Product IDBRC0823
Product classBioreference compound
CAS number26675-46-7
MW184.5
Synonyms
R-E 235da1, HCFE 235da2,
Transport conditionsNormal

Isoflurane

Isoflurane is a general inhalation anesthetic. It induces a reduction in junctional conductance by decreasing gap junction channel opening times and increasing gap junction channel closing times.

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BRC0687
Product IDBRC0687
Product classBioreference compound
CAS number13838-16-9
MW184.5
Synonyms
Anesthetic 347; Alyrane;
Transport conditionsNormal

Enflurane

Enflurane is an anesthetic. It induces muscle relaxation and reduces pains sensitivity by altering tissue excitability. Enflurane acts as a positive allosteric modulator of the GABAA, glycine, and 5-HT3 receptors, and as a negative allosteric modulator of the AMPA, kainate, and NMDA receptors, as well as of nicotinic acetylcholine receptors.

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BRC0857
Product IDBRC0857
Product classBioreference compound
CAS number28523-86-6
MW200.1
Synonyms
Transport conditionsNormal

Sevoflurane

Sevoflurane is one of the most commonly used volatile anesthetic agents, particularly for outpatient anesthesia, across all ages, as well as in veterinary medicine.

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BRC0814
Product IDBRC0814
Product classBioreference compound
CAS number15687-27-1
MW206.3
Synonyms
NSC 256857; U-18753;
Transport conditionsNormal

Ibuprofen

Ibuprofen is a nonsteroidal anti-inflammatory agent with analgesic and antipyretic properties. It is a non-selective, reversible COX inhibitor (IC50 for human recombinant COX-1 and COX-2 are 2.6 and 1.53 µM, respectively).

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BRC0827
Product IDBRC0827
Product classBioreference compound
CAS number51146-56-6
MW206.3
Synonyms
d-ibuproten; S(+)-ibuprofen;
Transport conditionsNormal

Dexibuprofen

Dexibuprofen is a non-steroidal anti-inflammatory drug. It is a pharmacologically effective enantiomer of racemic ibuprofen that differs in physicochemical properties.

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BRC0999
Product IDBRC0999
Product classBioreference compound
CAS number66-84-2
MW215.6
Synonyms
Chitosamine;
Transport conditionsNormal

Glucosamine Hydrochloride

Glucosamine is an amino sugar and a prominent precursor in the biochemical synthesis of glycosylated proteins and lipids.

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BRC0226
Product IDBRC0226
Product classBioreference compound
CAS number125-33-7
MW218.3
Synonyms
Desoxyphenobarbital, Mysoline, Liskantin, Mizodin, Mylepsinum, Pridona, Primid, Prysoline, Sertan
Transport conditionsNormal
Restrictions Included in DEA controlled list

Primidone

An antiepileptic agent related to the barbiturates; it is partly metabolized to phenobarbital in the body and owes some of its actions to this metabolite. Primidone is a GABA receptor agonist.

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BRC0445
Product IDBRC0445
Product classBioreference compound
CAS number33125-97-2
MW244.3
Synonyms
Lipuro, Propiscin, R 16659, Hypnomidate, Amidate
Transport conditionsNormal

Etomidate

Etomidate is an imidazole compound that appears to depress CNS function via GABA and categorized as an anesthetic. Etomidate also inhibits adrenal cortisol biosynthesis and mitigates hypercortisolism, as is found in Cushing syndrome.

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BRC1061
Product IDBRC1061
Product classBioreference compound
CAS number77191-36-7
MW246.3
Synonyms
DM 9384; DMMPA; DMPPA; DZL 221; Translon;
Transport conditionsNormal

Nefiracetam

Nefiracetam is cognitive enhancer that displays various pharmacological effects. Activates L/N-type calcium channels, cholinergic, monoaminergic and GABAergic systems. Displays potent neuroprotective action in the retinal ischemia-reperfusion model in vivo.

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BRC0246
Product IDBRC0246
Product classBioreference compound
CAS number28311-31-1
MW250.1
Synonyms
(+-)-Baclofen, Baclon, Kemstro, Lioresal Intrathecal,
Transport conditionsNormal

Baclofen hydrochloride

Baclofen is a direct agonist at GABAB receptors.

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BRC0045
Product IDBRC0045
Product classBioreference compound
CAS number78755-81-4
MW303.3
Synonyms
Anexate, Flumazepil, Romazicon, Lanexat, Ro 15-1788
Transport conditionsNormal

Flumazenil

Flumazenil antagonizes the CNS effects produced by benzodiazepines, but does not antagonize the central nervous system effects of drugs affecting GABA-ergic neurons by means other than the benzodiazepine receptor (including ethanol, barbiturates, or general anesthetics) and does not reverse the effects of opioids

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BRC0918
Product IDBRC0918
Product classBioreference compound
CAS number70-18-8
MW307.3
Synonyms
GSH; Isethion; L-Glutathione Reduced;
Transport conditionsNormal

Glutathione

Glutathione reduces reactive oxygen species formed during cellular metabolism. Regulates activity of the redox-sensitive transcription factor NF-κB. Glutathione participates in leukotriene synthesis and is a cofactor for the enzyme glutathione peroxidase.

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BRC0748
Product IDBRC0748
Product classBioreference compound
CAS number132539-06-1
MW312.4
Synonyms
ADAMED, Arenbil, Integrol, LY 170053
Transport conditionsNormal

Olanzapine

Olanzapine is serotonin (5-HT2) and dopamine (D1/D2) receptor antagonist with anticholinergic and antipsychotic activity.

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BRC0109
Product IDBRC0109
Product classBioreference compound
CAS number14028-44-5
MW313.8
Synonyms
Asendin, Demolox, CL 67772
Transport conditionsNormal
Restrictions Included in California Proposition 65 list  WARNING! This product contains a chemical known to the State of California to cause birth defects or other reproductive harm. For more information go to www.P65Warnings.ca.gov.

Amoxapine

Amoxapine is a tricyclic dibenzoxazepine (an N-aryl piperazine) which acts similarly to several other tricyclic antidepressants; amoxapine inhibits GLYT2a transport activity with IC50 of 92 M.

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BRC0634
Product IDBRC0634
Product classBioreference compound
CAS number220860-50-4
MW323.4
Synonyms
Transport conditionsNormal

CP 457920

CP 457920 is GABAA inverse agonist (Ki < 1 µM).

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BRC0184
Product IDBRC0184
Product classBioreference compound
CAS number97240-79-4
MW339.4
Synonyms
McN-4853, RWJ-17021, Topamax, TPM
Transport conditionsNormal
Restrictions Included in California Proposition 65 list  WARNING! This product contains a chemical known to the State of California to cause birth defects or other reproductive harm. For more information go to www.P65Warnings.ca.gov.

Topiramate

Topiramate is an anticonvulsant indicated in the treatment of epilepsy and migraine. Topiramate enhances GABA-activated chloride channels. In addition, topiramate inhibits excitatory neurotransmission, through actions on kainate and AMPA receptors. There is evidence that topiramate has a specific effect on GluR5 kainate receptors.

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BRC1060
Product IDBRC1060
Product classBioreference compound
CAS number94875-80-6
MW368.4
Synonyms
E100; INS-100(I); NSC-32982;
Transport conditionsNormal

Curcumin

Curcumin is a yellow-orange dye and possesses a vast number of biological targets. It is an antitumor, anti-inflammatory, and antioxidant agent.

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BRC0272
Product IDBRC0272
Product classBioreference compound
CAS number77337-73-6
MW400.5
Synonyms
N-acetyl homotaurine, N-Acetylhomotaurine, Campral, Regtect
Transport conditionsNormal

Acamprosate Calcium

Acamprosate Calcium is a GABA receptor agonist and modulator of glutamatergic systems.

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BRC0108
Product IDBRC0108
Product classBioreference compound
CAS number145821-59-6
MW412.0
Synonyms
Gabitril, NO050328, NO328, TGB
Transport conditionsNormal

Tiagabine hydrochloride

Tiagabine is an anti-convulsive medication. It is also used in the treatment for panic disorder as are a few other anticonvulsants. Though the exact mechanism by which tiagabine exerts its effect on the human body is unknown, it does appear to operate as a selective GABA reuptake inhibitor.

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BRC0656
Product IDBRC0656
Product classBioreference compound
CAS number1026822-49-0
MW421.8
Synonyms
Transport conditionsNormal

5-(4-chlorophenyl)-N-{[2-(2,2,2-trifluoroethoxy)pyridin-3-yl]methyl}pyridine-3-carboxamide

The compound is potent sodium channel protein type blocker (IC50 = 0.003 µM).

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BRC0280
Product IDBRC0280
Product classBioreference compound
CAS number70288-86-7
MW861.1
Synonyms
Ivermax, Ivomec, Mectizan, Noromectin, Privermectin, Sklice, Stromectol, Vetrimec, Zimecterin, MK933
Transport conditionsNormal

Ivermectin

Ivermectin is a semisynthetic, anthelminitic agent.

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