Other kinases
| Structure | Product info | Availability | Quantity / Price |
|---|---|---|---|
 | Product IDBRC1048 Product classBioreference compound CAS number62613-82-5 MW Synonyms CGP 21690; CT 848; Hydroxypiracetam; ISF 2522; Neuractiv; Transport conditionsNormal OxiracetamOxiracetam, a cyclic derivative of gamma-aminobutyric acid (GABA), is a nootropic drug of the racetam family and very mild stimulant. | In Stock(5 business days) |  |
 | Product IDBRC0168 Product classBioreference compound CAS number89-57-6 MW153.1 Synonyms 5-ASA, Asacol, Asacolitin, Canasa, Claversal, Fisalamine, Iialda, Lixacol, m-Aminosalicylic acid, P-Aminosalicylsaeure, Pentasa, Rowasa, Salofalk Transport conditionsNormal MesalazineAn anti-inflammatory agent, structurally related to the salicylates, which is active in inflammatory bowel disease. It is considered to be the active moiety of sulphasalazine. | In Stock(5 business days) | |
 | Product IDBRC1305 Product classBioreference compound CAS number68252-28-8 MW158.2 Synonyms Transport conditionsNormal (R)-(+)-Oxiracetam(R)-(+)-Oxiracetam is enantiomer of Oxiracetam, nootropic drug. | In Stock(5 business days) | |
 | Product IDBRC0148 Product classBioreference compound CAS number1115-70-4 MW165.6 Synonyms Glucophage, Dimethylbiguanide, Glumetza, Metiguanide Transport conditionsNormal Metformin hydrochlorideMetformin is an oral antihyperglycemic agent that improves glucose tolerance in patients with NIDDM, lowering both basal and postprandial plasma glucose. | In Stock(5 business days) | |
 | Product IDBRC1104 Product classBioreference compound CAS number459-86-9 MW184.2 Synonyms NSC 32946; MGBG; Transport conditionsNormal MitoguazoneMitoguazone is a drug used in chemotherapy, in trials studying the treatment of Lymphoma, HIV Infections, and Non-Hodgkin Lymphoma. | In Stock(5 business days) | |
 | Product IDBRC0628 Product classBioreference compound CAS number13721-01-2 MW189.2 Synonyms Transport conditionsNormal 4-Quinolone-3-carboxylic acid4-Quinolone-3-carboxylic acidis a novel HIV-1 integrase strand transfer inhibitor. | In Stock(5 business days) | |
 | Product IDBRC0150 Product classBioreference compound CAS number1313437-84-1 MW209.9 Synonyms Trilithium citrate Transport conditionsNormal Restrictions
Included in California Proposition 65 list
Restriction
WARNING! This product contains a chemical known to the State of California to cause health damage.
For more information go to
www.P65Warnings.ca.gov.
Lithium CitrateLithium salts such as lithium carbonate, lithium citrate, and lithium orotate are mood stabilizers. They are used in the treatment of bipolar disorder, since unlike most other mood altering drugs, they counteract both mania and depression. | In Stock(5 business days) | |
 | Product IDBRC0831 Product classBioreference compound CAS number59277-89-3 MW225.2 Synonyms NSC-645011, BW 248U Transport conditionsNormal AciclovirAciclovir is a synthetic deoxyguanosine analog and it is the prototype antiviral agent that is activated by viral thymidine kinase. | In Stock(5 business days) | |
 | Product IDBRC0233 Product classBioreference compound CAS number82410-32-0 MW255.2 Synonyms GA2, Cytovene, Vitrasert, RS-21592, BW-759 Transport conditionsNormal Restrictions
Included in California Proposition 65 list
Restriction
WARNING! This product contains a chemical known to the State of California to cause cancer and birth defects or other reproductive harm.
For more information go to
www.P65Warnings.ca.gov.
GanciclovirGanciclovir is a synthetic nucleoside analogue of 2'-deoxyguanosine that inhibits replication of herpes viruses both in vitro and in vivo. Ganciclovir is a prodrug that is structurally similar to acyclovir. | In Stock(5 business days) | |
 | Product IDBRC0771 Product classBioreference compound CAS number95058-81-4 MW263.2 Synonyms LY188011, NSC 613327, Zefei, DDFC Transport conditionsNormal GemcitabineGemcitabine is an antineoplastic anti-metabolite that inhibits DNA synthesis. | In Stock(5 business days) | |
 | Product IDBRC0243 Product classBioreference compound CAS number75706-12-6 MW270.2 Synonyms Arava, HW 486, Avara, SU 101 Transport conditionsNormal LeflunomideLeflunomide is a pyrimidine synthesis inhibitor indicated in adults for the treatment of active rheumatoid arthritis (RA). | In Stock(5 business days) | |
 | Product IDBRC0510 Product classBioreference compound CAS number327033-36-3 MW273.2 Synonyms TCS PIM-1 4a Transport conditionsNormal SMI-4aSMI-4a is a potent selective ATP-competitive Pim-1 kinase inhibitor with an IC50 of 21 nM for Pim-1 compared to an IC50 of 100 nM for Pim-2. Does not significantly inhibit any other serine/threonine- or tyrosine-kinases. | In Stock(5 business days) | |
 | Product IDBRC0514 Product classBioreference compound CAS number116970-50-4 MW287.8 Synonyms Protein kinase inhibitor H-9 Transport conditionsNormal H-9 hydrochlorideH-9 (hydrochloride), an isoquinolinesulfonamide protein kinase inhibitor, is a competitive inhibitor of PKC, PKG, and PKA with Ki values of 18, 0.87, and 1.9 µM, respectively. | In Stock(5 business days) | |
 | Product IDBRC0302 Product classBioreference compound CAS number103745-39-7 MW291.4 Synonyms ZK-258594, HA-1077, AT-877 Transport conditionsNormal FasudilFasudil is a class of calcium antagonists. Fasudil is able to inhibit contractile responses to KCl, phenylephnne (PHE) and prostaglandin (PG) F2a. Fasudil also exhibits vasodilator actions by inhibition of 5-hydroxytryptamine, noradrenaline, histamine, angiotensin, and dopamine induced spiral strips contraction | In Stock(5 business days) | |
 | Product IDBRC0667 Product classBioreference compound CAS number125314-13-8 MW317.3 Synonyms Transport conditionsNormal CP21R7CP21R7 is a potent and selective inhibitor of GSK3 beta (IC50 = 1.8 nM). | In Stock(5 business days) | |
 | Product IDBRC0743 Product classBioreference compound CAS number836620-48-5 MW347.4 Synonyms Transport conditionsNormal AS1842856AS1842856 is cell-permeable oxodihydroquinoline that preferentially inhibits the transcription activity of Forkhead box O family member Foxo1 (IC50 = 33 nM) over that of the functionally related Foxo3a and Foxo4 (70%, 20%, and 3% inhibition, respectively, in HepG2-based reporter assays) via direct binding of the active Foxo1, but not the Ser256-phosphorylated/inactive form of Foxo1. | In Stock(5 business days) | |
 | Product IDBRC0558 Product classBioreference compound CAS number301305-73-7 MW360.4 Synonyms Transport conditionsNormal TCS 359TCS 359 is a potent inhibitor of FLT3 receptor tyrosine kinase (IC50 = 42 nM) that displays selectivity over a range of other kinases. | In Stock(5 business days) | |
 | Product IDBRC0398 Product classBioreference compound CAS number124832-27-5 MW360.8 Synonyms Bagovir, Cycloval,Mitanga, Ovalac, Pervioral, Revira, Vacyless, Vadiral, Valdacir, Valotix, Valtrex, Valvir, Valztrex, Viramixal, Viropel, Vociflon, Zelitrex, Zelivire Transport conditionsNormal Valaciclovir hydrochlorideValaciclovir (INN) or Valacyclovir (USAN) is a prodrug and synthetic purine nucleoside analogue with inhibitory activity against herpes simplex virus types 1 (HSV-1), 2 (HSV-2), varicella-zoster virus (VZV), Epstein-Barr virus (EBV), and cytomegalovirus (CMV). | In Stock(5 business days) | |
 | Product IDBRC0349 Product classBioreference compound CAS number75607-67-9 MW365.2 Synonyms F-ara-A (NSC 312887) Phosphate, NSC-118218 Transport conditionsNormal Fludarabine phosphateFludarabine is a chemotherapy drug used in the treatment of chronic lymphocytic leukemia. It acts at DNA polymerase alpha, ribonucleotide reductase and DNA primase, results in the inhibition of DNA synthesis, and destroys the cancer cells. | In Stock(5 business days) | |
 | Product IDBRC0064 Product classBioreference compound CAS number10540-29-1 MW371.5 Synonyms Zemide, Ethanamine, ICI 46474 Transport conditionsNormal Restrictions
Included in California Proposition 65 list
Restriction
WARNING! This product contains a chemical known to the State of California to cause cancer.
For more information go to
www.P65Warnings.ca.gov.
TamoxifenTamoxifen is indicated for the treatment of metastatic breast cancer in women and men and ductal carcinoma in Situ. Tamoxifen is a nonsteroidal agent that binds to estrogen receptors (ER), inducing a conformational change in the receptor. This results in a blockage or change in the expression of estrogen dependent genes. The prolonged binding of tamoxifen to the nuclear chromatin of these results in reduced DNA polymerase activity, impaired thymidine utilization, blockade of estradiol uptake, and decreased estrogen response. | In Stock(5 business days) | |
 | Product IDBRC0680 Product classBioreference compound CAS number169590-42-5 MW381.4 Synonyms Eurocox, Medicoxib, SC 58635, Xilebao, YM 177 Transport conditionsNormal CelecoxibCelecoxib is a selective cyclooxygenase-2 (Cox-2) inhibitor (IC50 = 40 nM) with low sensitivity against Cox-1. Celecoxib is a non-steroidal anti-inflammatory drug (NSAID) used in the treatment of osteoarthritis, rheumatoid arthritis, acute pain, painful menstruation and menstrual symptoms. | In Stock(5 business days) | |
 | Product IDBRC0635 Product classBioreference compound CAS number256477-09-5 MW385.8 Synonyms Transport conditionsNormal UK-371804UK-371804 is a potent and selective inhibitor of urokinase-type plasmogen activator (uPA) (Ki=10 nM). Selectivity is 4000-fold versus tPA and 2700-fold versus plasmin. | In Stock(5 business days) | |
 | Product IDBRC0531 Product classBioreference compound CAS number1209784-87-1 MW389.5 Synonyms Transport conditionsNormal 2-[[[2-(4-Ethoxy-3-methoxyphenyl)-4-thiazolyl]methyl]thio]-4,6-pyrimidinediamineThe compound is deoxycytidine kinase inhibitor (IC50 = 1.12 μM). | In Stock(5 business days) | |
 | Product IDBRC0702 Product classBioreference compound CAS number599-79-1 MW398.4 Synonyms NSC 203730, NSC 667219, Reupirin, Azulfin, Benzosulfa Transport conditionsNormal Restrictions
Included in California Proposition 65 list
Restriction
WARNING! This product contains a chemical known to the State of California to cause cancer and birth defects or other reproductive harm.
For more information go to
www.P65Warnings.ca.gov.
SulfasalazineSulfasalazine is an anti-inflammatory (gastrointestinal). It is inhibitor of NF-κB activation. Inhibits in vitro growth of the human pancreatic cancer cell lines MIA PaCa-2 and PANC-1, and induces apoptosis in glioblastoma cell lines. Also inhibits the cystine-glutamate antiporter, system Xc (SXC). | In Stock(5 business days) | |
 | Product IDBRC0502 Product classBioreference compound CAS number2060523-50-2 MW409.7 Synonyms Transport conditionsNormal 4-(aminomethyl)-N'-(5-bromo-2-oxo-2,3-dihydro-1H-indol-3-ylidene)benzohydrazide hydrochlorideIs an inhibitor of human recombinant PKR autophosphorylation. | In Stock(5 business days) | |
 | Product IDBRC0577 Product classBioreference compound CAS number1809862-74-5 MW424.5 Synonyms Transport conditionsNormal 3-methyloxetan-3-yl 4-[3-(2-methoxypyridin-3-yl)pyrazolo[1,5-a]pyrimidin-5-yl]piperazine-1-carboxylateThe compound is potent, brain penetrant inhibitor of AP2-associated protein kinase 1 (IC50 = 4.7 nM). | In Stock(5 business days) | |
 | Product IDBRC0331 Product classBioreference compound CAS number183319-69-9 MW429.9 Synonyms CP358774, NSC 718781 Transport conditionsNormal Erlotinib hydrochlorideErlotinib inhibits the intracellular phosphorylation of tyrosine kinase associated with the epidermal growth factor receptor (EGFR). | In Stock(5 business days) | |
 | Product IDBRC0376 Product classBioreference compound CAS number1042432-58-5 MW438.9 Synonyms Transport conditionsNormal CTx-0152960CTx-0152960, was reported as a new member of the broad spectrum PKI family and developed as a Sepharose-supported kinase capture reagent in the identification of 235 protein kinases from a digest of human breast adenocarcinoma, MDA-MB-231, cells. | In Stock(5 business days) | |
 | Product IDBRC0592 Product classBioreference compound CAS number1448694-02-7 MW447.5 Synonyms Transport conditionsNormal GCN2-IN-3GCN2-IN-3 is inhibitor of GCN2 (IC50 < 0.3 µM). | In Stock(5 business days) | |
 | Product IDBRC0723 Product classBioreference compound CAS number1589527-65-0 MW518.5 Synonyms Transport conditionsNormal KIRA 6KIRA 6 is an allosteric inhibitor of IRE1α RNase, preserves cell viability and function in ER-stressed retinitis pigmentosa and diabetes model cells. | In Stock(5 business days) | |
 | Product IDBRC0332 Product classBioreference compound CAS number388082-78-8 MW581.1 Synonyms FMM, GW 572016, Tykerb Transport conditionsNormal Lapatinib ditosylateLapatinib is a 4-anilinoquinazoline kinase inhibitor of the intracellular tyrosine kinase domains of both epidermal growth factor receptor (HER1/EGFR/ERBB1) and human epidermal growth factor receptor type 2 (HER2/ERBB2)with a dissociation half-life of ≥300 minutes. Lapatinib inhibits ERBB-driven tumor cell growth in vitro and in various animal models. | In Stock(5 business days) | |
 | Product IDBRC0255 Product classBioreference compound CAS number34031-32-8 MW678.5 Synonyms Ridaura, Triethylphosphine gold Transport conditionsNormal Restrictions
Included in California Proposition 65 list
Restriction
WARNING! This product contains a chemical known to the State of California to cause birth defects or other reproductive harm.
For more information go to
www.P65Warnings.ca.gov.
AuranofinAuranofin is a gold salt used in treating inflammatory arthritis. It may act as an inhibitor of kappab kinase and thioredoxin reductase which would lead to a decreased immune response and decreased free radical production, respectively. | In Stock(5 business days) | |