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Mitogen-activated protein kinase (MAPK)

StructureProduct infoAvailabilityQuantity / Price
BRC1044
Product IDBRC1044
Product classBioreference compound
CAS number61-80-3
MW168.6
Synonyms
Flexin; McN-485; NSC 24995; Zoxamin;
Transport conditionsNormal

Zoxazolamine

Zoxazolamine is a potent skeletal muscle relaxant that also has uricosuric activity. It is used as a tool for assessing hepatic cytochrome P-450 activity.

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BRC0476
Product IDBRC0476
Product classBioreference compound
CAS number315694-89-4
MW276.3
Synonyms
Transport conditionsNormal

TC-DAPK 6

TC-DAPK 6 is potent and selective, ATP-competitive inhibitor of death-associated protein kinase 1 (DAPK1) (IC50 values are 69 and 225 nM for DAPK1 and DAPK3 respectively, when assayed with 10 μM ATP). Displays selectivity for DAPK1 over a range of 48 other kinases, including Abl, AMPK, Chk1, Met and Src (IC50 > 10 μM).

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BRC0556
Product IDBRC0556
Product classBioreference compound
CAS number325979-58-6
MW300.4
Synonyms
Transport conditionsNormal

SB-347804

SB-347804 is a potent and selective inhibitor of JNK3 kinase (IC50 = 3.16 μM).

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BRC0340
Product IDBRC0340
Product classBioreference compound
CAS number794510-70-6
MW301.2
Synonyms
Transport conditionsNormal

ETP-45835

Mnk2 and Mnk1 inhibitor (IC50 values are 575 and 646 nM respectively). Exhibits selectivity against a panel of 24 protein kinases, including those upstream of Mnk1/2.

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BRC0472
Product IDBRC0472
Product classBioreference compound
CAS number380491-32-7
MW330.4
Synonyms
SJ000170251
Transport conditionsNormal

GNF-Pf-2466

GNF-Pf-2466 is kinase inhibitor. Also potential antitubercular agent (TB IC90 = 3.2).

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BRC0498
Product IDBRC0498
Product classBioreference compound
CAS number326886-05-9
MW355.2
Synonyms
Sulfonylhydrazone-
Transport conditionsNormal

Shz-1

Shz-1 is an activator of early cardiac genes (including Nkx2.5) in pluripotent stem cells. Induces phenotypic differentiation in human mobilized peripheral blood mononuclear cells. Enhances myocardial regenerative repair by stem cells in a rat myocardial cryoinjury model.

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BRC0793
Product IDBRC0793
Product classBioreference compound
CAS number710323-58-3
MW356.2
Synonyms
GSK 3 Inhibitor IX; MLS 2052; 6-Bromoindirubin-3-oxime;
Transport conditionsNormal

BIO

BIO is a cell-permeable, highly potent, selective, reversible and ATP-competitive glycogen synthase kinase-3 inhibitor. Maintains self-renewal and pluripotency in embryonic stem cells via activation of the Wnt signaling pathway in vitro. Also, promotes proliferation and dedifferentiation in cardiomyocytes.

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BRC0754
Product IDBRC0754
Product classBioreference compound
CAS number602293-00-5
MW419.5
Synonyms
Transport conditionsNormal

N-(3-Acetylphenyl)-9-amino-2,3-dihydro-1,4-dioxino[2,3-g]thieno[2,3-b]quinoline-8-carboxamide

The compound is a novel disruptor of the PKCε/RACK2 protein-protein interaction.

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BRC0442
Product IDBRC0442
Product classBioreference compound
CAS number924198-81-2
MW451.5
Synonyms
A17(SMURF1 inhibitor)
Transport conditionsNormal

A17

A17 is an inhibitor of ubiquitin ligase Smad ubiquitination regulatory factor-1 (Smuf1) that is a major regulator of bone morphogenetic protein (BMP) signaling. A17 strongly inhibits Smad1/5 ubiquitination mediated by Smuf1, increases BMP signal responsiveness and enhances BMP-2 induced osteoblastic activity.

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BRC0921
Product IDBRC0921
Product classBioreference compound
CAS number1007647-73-5
MW512.9
Synonyms
Transport conditionsNormal

A01 (Smurf1 inhibitor)

A01 is an inhibitor of ubiquitin ligase Smad ubiquitination regulatory factor-1 (Smuf1) that is a major regulator of bone morphogenetic protein (BMP) signaling. AO1 strongly inhibits Smad1/5 ubiquitination mediated by Smuf1, increases BMP signal responsiveness and enhances BMP-2 induced osteoblastic activity.

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BRC0434
Product IDBRC0434
Product classBioreference compound
CAS number1347797-73-2
MW1005.2
Synonyms
Transport conditionsNormal

calcium (3R,5R)-7-(4-(4-fluorophenyl)-6-isopropyl-2-(N-methylmethylsulfonamido)pyrimidin-5-yl)-3,5-dihydroxyheptanoate

Is rosuvastatin enantiomer compound that inhibits hydroxymethylglutaryl-coenzyme A (HMG-CoA) reductase, also has inhibitory activity against human recombinant p38 MAP kinase expressed in Escherichia coli using myelin basic protein (MBP).

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