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StructureProduct infoAvailabilityQuantity / Price
BRC1048
Product IDBRC1048
Product classBioreference compound
CAS number62613-82-5
MW
Synonyms
CGP 21690; CT 848; Hydroxypiracetam; ISF 2522; Neuractiv;
Transport conditionsNormal

Oxiracetam

Oxiracetam, a cyclic derivative of gamma-aminobutyric acid (GABA), is a nootropic drug of the racetam family and very mild stimulant.

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BRC1316
Product IDBRC1316
Product classBioreference compound
CAS number328-50-7
MW146.1
Synonyms
NSC 17391; 2-Ketoglutaric acid;
Transport conditionsNormal

2-Oxoglutaric acid

2-Oxoglutaric acid is an intermediate in the Krebs cycle catalyzed by glutamate dehydrogenase enzyme on glutamate.

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BRC0168
Product IDBRC0168
Product classBioreference compound
CAS number89-57-6
MW153.1
Synonyms
5-ASA, Asacol, Asacolitin, Canasa, Claversal, Fisalamine, Iialda, Lixacol, m-Aminosalicylic acid, P-Aminosalicylsaeure, Pentasa, Rowasa, Salofalk
Transport conditionsNormal

Mesalazine

An anti-inflammatory agent, structurally related to the salicylates, which is active in inflammatory bowel disease. It is considered to be the active moiety of sulphasalazine. 

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BRC0194
Product IDBRC0194
Product classBioreference compound
CAS number65-49-6
MW153.1
Synonyms
PAS, Mesalamine
Transport conditionsNormal

4-Aminosalicylic Acid

Aminosalicylic acid is an anti-mycobacterial agent used with other anti-tuberculosis drugs (most often isoniazid) for the treatment of all forms of active tuberculosis due to susceptible strains of tubercle bacilli.

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BRC1305
Product IDBRC1305
Product classBioreference compound
CAS number68252-28-8
MW158.2
Synonyms
Transport conditionsNormal

(R)-(+)-Oxiracetam

(R)-(+)-Oxiracetam is enantiomer of Oxiracetam, nootropic drug.

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BRC0818
Product IDBRC0818
Product classBioreference compound
CAS number616-91-1
MW163.2
Synonyms
5052; NSC-111180; RK-0202; NAC; Mercapturic acid;
Transport conditionsNormal

Acetylcysteine

Acetylcysteine (NAC) is an antioxidant and precursor of glutathione that has multiple effects in cells and animals. It is primarily used as a mucolytic agent and in the management of acetaminophen poisoning. It is essentially a prodrug that is converted to cysteine (in the intestine by the enzyme aminoacylase 1) and absorbed in the intestine into the bloodstream. As an antioxidant, NAC scavenges hydrogen peroxide, hydroxyl radical, and hypochlorous acid.

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BRC0148
Product IDBRC0148
Product classBioreference compound
CAS number1115-70-4
MW165.6
Synonyms
Glucophage, Dimethylbiguanide, Glumetza, Metiguanide
Transport conditionsNormal

Metformin hydrochloride

Metformin is an oral antihyperglycemic agent that improves glucose tolerance in patients with NIDDM, lowering both basal and postprandial plasma glucose.

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BRC1044
Product IDBRC1044
Product classBioreference compound
CAS number61-80-3
MW168.6
Synonyms
Flexin; McN-485; NSC 24995; Zoxamin;
Transport conditionsNormal

Zoxazolamine

Zoxazolamine is a potent skeletal muscle relaxant that also has uricosuric activity. It is used as a tool for assessing hepatic cytochrome P-450 activity.

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BRC0936
Product IDBRC0936
Product classBioreference compound
CAS number50-78-2
MW180.2
Synonyms
BAY1019036; NSC-27223; NSC-406186; ASA; Aspirin;
Transport conditionsNormal
Restrictions Included in California Proposition 65 list Restriction  WARNING! This product contains a chemical known to the State of California to cause birth defects or other reproductive harm. For more information go to www.P65Warnings.ca.gov.

Acetylsalicylic acid

Acetylsalicylic acid is an anti-inflammatory and antipyretic agent and acts as the inhibitor of cyclooxygenase which results in the inhibition of the biosynthesis of prostaglandins. It also inhibits platelet aggregation and is used in the prevention of arterial and venous thrombosis.

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BRC1104
Product IDBRC1104
Product classBioreference compound
CAS number459-86-9
MW184.2
Synonyms
NSC 32946; MGBG;
Transport conditionsNormal

Mitoguazone

Mitoguazone is a drug used in chemotherapy, in trials studying the treatment of Lymphoma, HIV Infections, and Non-Hodgkin Lymphoma.

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BRC0628
Product IDBRC0628
Product classBioreference compound
CAS number13721-01-2
MW189.2
Synonyms
Transport conditionsNormal

4-Quinolone-3-carboxylic acid

4-Quinolone-3-carboxylic acidis a novel HIV-1 integrase strand transfer inhibitor.

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BRC0452
Product IDBRC0452
Product classBioreference compound
CAS number1485-00-3
MW193.2
Synonyms
NSC 10120, NSC 105303, NSC 170724, Syk Inhibitor III
Transport conditionsNormal

MNS

MNS is selective inhibitor of Src and Syk tyrosine kinases. Displays antiaggregative activity via inhibition of GPIIb/IIIa activation (IC50 = 12.7 μM for thrombin-induced platelet aggregation). Exhibits no effects on Ca2+-dependent enzymes, PKC or arachidonic acid metabolism.

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BRC0295
Product IDBRC0295
Product classBioreference compound
CAS number58-08-2
MW194.2
Synonyms
Methyltheobromine, NSC 5036
Transport conditionsNormal

Caffeine

Central nervous system stimulant. Antagonist at A1 and A2A adenosine receptors and inhibitor of cyclic nucleotide phosphodiesterases. Mobilizes calcium from intracellular stores and inhibits benzodiazepine binding to GABA receptors.

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BRC0365
Product IDBRC0365
Product classBioreference compound
CAS number15421-84-8
MW205.3
Synonyms
Rocornal, Trapymin, Avantrin, Trapymine
Transport conditionsNormal

Trapidil

Trapidil interrupts the autocrine loop at the PDGF and PDGF-receptor level.Trapidil has proved to possess a significant antiproliferative activity. Trapidil is an anti-platelet drug active against various aggregating agents, such as collagen, ADP, arachidonic acid, PAF and calcium ionophore.

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BRC0150
Product IDBRC0150
Product classBioreference compound
CAS number1313437-84-1
MW209.9
Synonyms
Trilithium citrate
Transport conditionsNormal
Restrictions Included in California Proposition 65 list Restriction  WARNING! This product contains a chemical known to the State of California to cause health damage. For more information go to www.P65Warnings.ca.gov.

Lithium Citrate

Lithium salts such as lithium carbonate, lithium citrate, and lithium orotate are mood stabilizers. They are used in the treatment of bipolar disorder, since unlike most other mood altering drugs, they counteract both mania and depression.

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BRC0609
Product IDBRC0609
Product classBioreference compound
CAS number776-53-4
MW213.3
Synonyms
Transport conditionsNormal

NSC 9310

NSC 9310 is CDK inhibitor.

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BRC0580
Product IDBRC0580
Product classBioreference compound
CAS number773-76-2
MW214.0
Synonyms
Endiaron; NSC 3904; Quesyl; CHQ;
Transport conditionsNormal

Chloroxine

Chloroxine is a synthetic antibacterial compound. It inhibits the growth of gram-positive as well as some gram-negative organisms.

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BRC0300
Product IDBRC0300
Product classBioreference compound
CAS number129-56-6
MW220.2
Synonyms
Nsc75890,
Transport conditionsNormal

SP600125

SP600125 is an anthrapyrazolone inhibitor of JNK that competes with ATP to inhibit the phosphorylation of c-Jun. It prevents the activation of inflammatory genes such as COX-2, IL-2 IFN-γ and TNF-α.8,9 It prevents the activation of JNK after brain ischemia and may be effective in treatment of ischemic stroke.

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BRC0831
Product IDBRC0831
Product classBioreference compound
CAS number59277-89-3
MW225.2
Synonyms
NSC-645011, BW 248U
Transport conditionsNormal

Aciclovir

Aciclovir is a synthetic deoxyguanosine analog and it is the prototype antiviral agent that is activated by viral thymidine kinase.

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BRC0877
Product IDBRC0877
Product classBioreference compound
CAS number2447-23-6
MW229.1
Synonyms
Transport conditionsNormal

SNX9-1

SNX9-1 is a CDK inhibitor.

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BRC0630
Product IDBRC0630
Product classBioreference compound
CAS number71897-07-9
MW234.3
Synonyms
AG-1295, NSC 380341
Transport conditionsNormal

Tyrphostin AG-1295

Tyrphostin AG 1295 is a cell-permeable, reversible, ATP-competitive and selective inhibitor of PDGFR (platelet-derived growth factor receptor) protein tyrosine kinase (PDGF-receptor PTK)(IC50 = 500 nM) and PDGF-dependent DNA synthesis (IC50 = 2.5 μM) in Swiss/3T3 cells, and demonstrates about 50% inhibition on neointimal formation after balloon injury in porcine femoral arteries.

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BRC0082
Product IDBRC0082
Product classBioreference compound
CAS number51-30-9
MW247.7
Synonyms
Norisodrine, Novodrin, Isopropydrin, Aludrine
Transport conditionsNormal

Isoproterenol hydrochloride

Isoproterenol is a relatively selective beta2-adrenergic bronchodilator. Isoproterenol is indicated for the relief of bronchospasm associated with chronic obstructive pulmonary disease.

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BRC0947
Product IDBRC0947
Product classBioreference compound
CAS number68-35-9
MW250.3
Synonyms
Adiazine;
Transport conditionsNormal

Sulfadiazine

Sulfadiazine is a sulfonamide antibiotic with a wide spectrum against most gram-positive and many gram-negative organisms. It is a competitive inhibitor of the bacterial enzyme dihydropteroate synthetase.

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BRC0233
Product IDBRC0233
Product classBioreference compound
CAS number82410-32-0
MW255.2
Synonyms
GA2, Cytovene, Vitrasert, RS-21592, BW-759
Transport conditionsNormal
Restrictions Included in California Proposition 65 list Restriction  WARNING! This product contains a chemical known to the State of California to cause cancer and birth defects or other reproductive harm. For more information go to www.P65Warnings.ca.gov.

Ganciclovir

Ganciclovir is a synthetic nucleoside analogue of 2'-deoxyguanosine that inhibits replication of herpes viruses both in vitro and in vivo. Ganciclovir is a prodrug that is structurally similar to acyclovir.

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BRC0121
Product IDBRC0121
Product classBioreference compound
CAS number50-35-1
MW258.2
Synonyms
Thalomid, Distaval, Softenon, Talimol,
Transport conditionsNormal
Restrictions Included in California Proposition 65 list Restriction  WARNING! This product contains a chemical known to the State of California to cause birth defects or other reproductive harm. For more information go to www.P65Warnings.ca.gov.

Thalidomide

Thalidomide is an immunomodulatory agent with a spectrum of activity that is not fully characterized. Thalidomide is racemic — it contains both left and right handed isomers in equal amounts: one enantiomer is effective against morning sickness, and the other is teratogenic.

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BRC0771
Product IDBRC0771
Product classBioreference compound
CAS number95058-81-4
MW263.2
Synonyms
LY188011, NSC 613327, Zefei, DDFC
Transport conditionsNormal

Gemcitabine

Gemcitabine is an antineoplastic anti-metabolite that inhibits DNA synthesis.

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BRC1295
Product IDBRC1295
Product classBioreference compound
CAS number51298-62-5
MW269.7
Synonyms
Transport conditionsNormal

L-NAME hydrochloride

L-NAME hydrochloride is a nonselective inhibitor of nitric oxide synthetases.

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BRC0243
Product IDBRC0243
Product classBioreference compound
CAS number75706-12-6
MW270.2
Synonyms
Arava, HW 486, Avara, SU 101
Transport conditionsNormal

Leflunomide

Leflunomide is a pyrimidine synthesis inhibitor indicated in adults for the treatment of active rheumatoid arthritis (RA).

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BRC0503
Product IDBRC0503
Product classBioreference compound
CAS number22816-60-0
MW271.6
Synonyms
Transport conditionsNormal

A 22 hydrochloride

A22 s a cell-permeable isothiourea compound that inhibits MreB, an actin-like bacterial protein, and has been shown to act as an antiobiotic adjuvant.

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BRC0510
Product IDBRC0510
Product classBioreference compound
CAS number327033-36-3
MW273.2
Synonyms
TCS PIM-1 4a
Transport conditionsNormal

SMI-4a

SMI-4a is a potent selective ATP-competitive Pim-1 kinase inhibitor with an IC50 of 21 nM for Pim-1 compared to an IC50 of 100 nM for Pim-2. Does not significantly inhibit any other serine/threonine- or tyrosine-kinases.

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BRC0476
Product IDBRC0476
Product classBioreference compound
CAS number315694-89-4
MW276.3
Synonyms
Transport conditionsNormal

TC-DAPK 6

TC-DAPK 6 is potent and selective, ATP-competitive inhibitor of death-associated protein kinase 1 (DAPK1) (IC50 values are 69 and 225 nM for DAPK1 and DAPK3 respectively, when assayed with 10 μM ATP). Displays selectivity for DAPK1 over a range of 48 other kinases, including Abl, AMPK, Chk1, Met and Src (IC50 > 10 μM).

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BRC0514
Product IDBRC0514
Product classBioreference compound
CAS number116970-50-4
MW287.8
Synonyms
Protein kinase inhibitor H-9
Transport conditionsNormal

H-9 hydrochloride

H-9 (hydrochloride), an isoquinolinesulfonamide protein kinase inhibitor, is a competitive inhibitor of PKC, PKG, and PKA with Ki values of 18, 0.87, and 1.9 µM, respectively.

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BRC0302
Product IDBRC0302
Product classBioreference compound
CAS number103745-39-7
MW291.4
Synonyms
ZK-258594, HA-1077, AT-877
Transport conditionsNormal

Fasudil

Fasudil is a class of calcium antagonists. Fasudil is able to inhibit contractile responses to KCl, phenylephnne (PHE) and prostaglandin (PG) F2a. Fasudil also exhibits vasodilator actions by inhibition of 5-hydroxytryptamine, noradrenaline, histamine, angiotensin, and dopamine induced spiral strips contraction

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BRC0556
Product IDBRC0556
Product classBioreference compound
CAS number325979-58-6
MW300.4
Synonyms
Transport conditionsNormal

SB-347804

SB-347804 is a potent and selective inhibitor of JNK3 kinase (IC50 = 3.16 μM).

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BRC0340
Product IDBRC0340
Product classBioreference compound
CAS number794510-70-6
MW301.2
Synonyms
Transport conditionsNormal

ETP-45835

Mnk2 and Mnk1 inhibitor (IC50 values are 575 and 646 nM respectively). Exhibits selectivity against a panel of 24 protein kinases, including those upstream of Mnk1/2.

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BRC0303
Product IDBRC0303
Product classBioreference compound
CAS number117-39-5
MW302.2
Synonyms
Sophoretin, Meletin, Quercetol, Xanthaurine
Transport conditionsNormal

Quercetin

Quercetin is a type of plant-based chemical. In several studies, it may have anti-inflammatory and antioxidant properties, and it is being investigated for a wide range of potential health benefits. Quercetin is a PI3K inhibitor with IC50 of 2.4 – 5.4 μM.

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BRC1032
Product IDBRC1032
Product classBioreference compound
CAS number521-74-4
MW303.0
Synonyms
Fenilor; Intensopan; NSC 1810; NSC 74937;
Transport conditionsNormal

Broxyquinoline

Broxyquinoline is an antiprotozoal agent.

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BRC0545
Product IDBRC0545
Product classBioreference compound
CAS number330786-24-8
MW303.3
Synonyms
Transport conditionsNormal

3-(4-Phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine

The compound is a highly selective Bruton’s tyrosine kinase (BTK) irreversible inhibitor (IC50 < 10 µM) and useful synthetic intermediate in the synthesis of Ibrutinib.

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BRC0433
Product IDBRC0433
Product classBioreference compound
CAS number154447-36-6
MW307.3
Synonyms
NSC 697286, SF 1101, LY 294002
Transport conditionsNormal

LY294002

LY294002 is a potent inhibitor of numerous proteins, and a strong inhibitor of phosphoinositide 3-kinases (PI3Ks).

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BRC0667
Product IDBRC0667
Product classBioreference compound
CAS number125314-13-8
MW317.3
Synonyms
Transport conditionsNormal

CP21R7

CP21R7 is a potent and selective inhibitor of GSK3 beta (IC50 = 1.8 nM).

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BRC0343
Product IDBRC0343
Product classBioreference compound
CAS number50264-69-2
MW321.2
Synonyms
AF 1890, Diclondazolic Acid
Transport conditionsNormal

Lonidamine

Anticancer and antispermatogenic agent in vitro and in vivo. Inhibits cellular energy metabolism in some cells via inhibition of mitochondrial hexokinase. Also blocks CFTR Cl- channels in vitro.

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BRC1405
Product IDBRC1405
Product classBioreference compound
CAS number5545-17-5
MW324.4
Synonyms
N,N-Diacetyl-L-cystine; NSC 203780; D-7193; DiNAC;
Transport conditionsNormal

N,N-Diacetylcystine

N,N-Diacetylcystine is an immunosuppressant potentially for the treatment of asthma.

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BRC0472
Product IDBRC0472
Product classBioreference compound
CAS number380491-32-7
MW330.4
Synonyms
SJ000170251
Transport conditionsNormal

GNF-Pf-2466

GNF-Pf-2466 is kinase inhibitor. Also potential antitubercular agent (TB IC90 = 3.2).

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BRC0480
Product IDBRC0480
Product classBioreference compound
CAS number329907-28-0
MW330.4
Synonyms
Transport conditionsNormal

TTP 22

TTP 22 is a high affinity casein kinase 2 (CK2) inhibitor (IC50 = 100 nM). Displays no inhibitory effects at 10 μM over JNK3, ROCK1, and MET.

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BRC0495
Product IDBRC0495
Product classBioreference compound
CAS number1347407-78-6
MW338.4
Synonyms
Transport conditionsNormal

4-{1H-pyrrolo[2,3-b]pyridin-3-yl}-N-[(thiophen-3-yl)methyl]-1,2,3,6-tetrahydropyridine-1-carboxamide

Rho-kinase inhibitor (IC50 = 10 μM).

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BRC0838
Product IDBRC0838
Product classBioreference compound
CAS number56296-78-7
MW345.8
Synonyms
Lilly 103472; Lilly 110 140; Prozac;
Transport conditionsNormal

Fluoxetine Hydrochloride

Fluoxetine hydrochloride is the first-in-class antidepressant, selective serotonin-reuptake inhibitor. It displays a selectivity for the serotonin transporter (Kd = 0.81 nM) over the norepinephrine transporter (Kd = 240 nM) and the dopamine transporter (Kd = 3,600 nM). It is used in the clinical treatment of major depression as well as other psychiatric disorders.

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BRC0743
Product IDBRC0743
Product classBioreference compound
CAS number836620-48-5
MW347.4
Synonyms
Transport conditionsNormal

AS1842856

AS1842856 is cell-permeable oxodihydroquinoline that preferentially inhibits the transcription activity of Forkhead box O family member Foxo1 (IC50 = 33 nM) over that of the functionally related Foxo3a and Foxo4 (70%, 20%, and 3% inhibition, respectively, in HepG2-based reporter assays) via direct binding of the active Foxo1, but not the Ser256-phosphorylated/inactive form of Foxo1.

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BRC0575
Product IDBRC0575
Product classBioreference compound
CAS number218156-96-8
MW349.4
Synonyms
Transport conditionsNormal

SRPIN340

SRPIN 340 is selective serine arginine protein kinase (SRPK) 1 inhibitor (Ki = 0.89 μM). Inhibits SRPK2 at higher concentrations. SRPIN 340 is competitive with ATP and does not inhibit other SRPKs significantly.

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BRC0574
Product IDBRC0574
Product classBioreference compound
CAS number848057-98-7
MW354.3
Synonyms
MVRL1
Transport conditionsNormal

SPHINX

SPHINX is SRPK1 kinase inhibitor (IC50 = 440 nM).

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BRC0498
Product IDBRC0498
Product classBioreference compound
CAS number326886-05-9
MW355.2
Synonyms
Sulfonylhydrazone-
Transport conditionsNormal

Shz-1

Shz-1 is an activator of early cardiac genes (including Nkx2.5) in pluripotent stem cells. Induces phenotypic differentiation in human mobilized peripheral blood mononuclear cells. Enhances myocardial regenerative repair by stem cells in a rat myocardial cryoinjury model.

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