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Antipsychotics

StructureProduct infoAvailabilityQuantity / Price
BRC0020
Product IDBRC0020
Product classBioreference compound
CAS number1986-47-6
MW169.6
Synonyms
Parnate; Transamine; Jatrosom;
Transport conditionsNormal

(1R,2S)-(+)-Tranylcypromine hydrochloride

Tranylcypromine hydrochloride is a non-hydrazine monoamine oxidase inhibitor with a rapid onset of activity.

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BRC1030
Product IDBRC1030
Product classBioreference compound
CAS number92-84-2
MW199.3
Synonyms
Fenoverm; NSC 2037; Dibenzothiazine; ENT 38;
Transport conditionsNormal

Phenothiazine

Phenothiazine is a rigid, tricyclic thiazine useful as an electron donor. It was formerly used as an insecticide and as a drug to treat infections with parasitic worms (anthelminthic).

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BRC0150
Product IDBRC0150
Product classBioreference compound
CAS number1313437-84-1
MW209.9
Synonyms
Trilithium citrate
Transport conditionsNormal
Restrictions Included in California Proposition 65 list  WARNING! This product contains a chemical known to the State of California to cause health damage. For more information go to www.P65Warnings.ca.gov.

Lithium Citrate

Lithium salts such as lithium carbonate, lithium citrate, and lithium orotate are mood stabilizers. They are used in the treatment of bipolar disorder, since unlike most other mood altering drugs, they counteract both mania and depression.

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BRC0004
Product IDBRC0004
Product classBioreference compound
CAS number145108-58-3
MW236.7
Synonyms
Precedex, Dex, Dexmedetomidine HCL, (S)-Medetomidine hydrochloride
Transport conditionsNormal

Dexmedetomidine hydrochloride

Dexmedetomidine (hydrochloride) is the (S)-enantiomer of medetomidine (racemic form of this compound), a highly selective, potent and specific agonist of 2-adrenergic receptor (2-adrenoceptor).

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BRC0107
Product IDBRC0107
Product classBioreference compound
CAS number196597-26-9
MW259.3
Synonyms
Rozerem, TAK-375
Transport conditionsNormal

Ramelteon

Ramelteon is a novel melatonin receptor agonist for human MT1 and MT2 receptors and chick forebrain melatonin receptors with Ki of 14 pM, 112 pM and 23.1 pM, respectively. Ramelteon is a melatonin receptor agonist with both high affinity for melatonin MT1 and MT2 receptors, and lower selectivity for the MT3 receptor.

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BRC0421
Product IDBRC0421
Product classBioreference compound
CAS number85650-52-8
MW265.4
Synonyms
Org 3770, 6-Azamianserin, Avanza, Axit, Mirtabene, Mirtaz, Mirtazon, Norset, Promyrtil, Remergil, Remergon, Remeron, Remeron SolTab, Rexer, Zispin
Transport conditionsNormal

Mirtazapine

Mirtazapine, an antidepressant of the piperazinoazepine class, is a tetracyclic compound with an anxiolytic effect. Mirtazapine has fewer ADRs than tricyclic antidepressants and is better tolerated. Selective blockade of specific serotonin receptors by mirtazapine likey minimizes side effects typical of other antidepressants.

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BRC0348
Product IDBRC0348
Product classBioreference compound
CAS number7416-34-4
MW276.4
Synonyms
Moban
Transport conditionsNormal

Molindone

An indole derivative effective in schizophrenia and other psychoses and possibly useful in the treatment of the aggressive type of undersocialized conduct disorder.

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BRC0403
Product IDBRC0403
Product classBioreference compound
CAS number99300-78-4
MW313.9
Synonyms
Elafax, Effexor, Efexor, Wy 45030
Transport conditionsNormal

Venlafaxine hydrochloride

Venlafaxine potentiates the neurotransmitter activity in the central nervous system. Furthermore, venlafaxine and its metabolite, O-desmethylvenlafaxine (ODV) potently inhibit the reuptake of serotonin and norepinephrine and weakly inhibit dopamine reuptake.

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BRC0360
Product IDBRC0360
Product classBioreference compound
CAS number113-59-7
MW315.9
Synonyms
NSC 169899
Transport conditionsNormal

Chlorprothixene

Chlorprothixene is a typical antipsychotic drug of the thioxanthene (tricyclic) class. Chlorprothixene exerts strong blocking effects by blocking the 5-HT2 D1, D2, D3, histamine H1, muscarinic and alpha1 adrenergic receptors.

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BRC0385
Product IDBRC0385
Product classBioreference compound
CAS number53-60-1
MW320.9
Synonyms
Sparine, Talofen
Transport conditionsNormal

Promazine hydrochloride

Promazine belongs to a group of medications known as the phenothiazine antipsychotics. It acts by blocking a variety of receptors in the brain, particularly dopamine receptors.

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BRC0997
Product IDBRC0997
Product classBioreference compound
CAS number15676-16-1
MW341.4
Synonyms
Transport conditionsNormal

Sulpiride

Sulpiride is selective dopamine D2 antagonist with antipsychotic and antidepressant activity.

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BRC0291
Product IDBRC0291
Product classBioreference compound
CAS number69-09-0
MW355.3
Synonyms
Chlorpromanyl, Largactil, Thorazine, J2.794D, NSC-167745, NSC-226514
Transport conditionsNormal

Chlorpromazine

Chlorpromazine is a psychotropic agent indicated for the treatment of schizophrenia. It antagonizes a range of receptors, including post-synaptic dopamine and serotonin receptors.

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BRC0608
Product IDBRC0608
Product classBioreference compound
CAS number1187159-50-7
MW360.5
Synonyms
Transport conditionsNormal

1-(2-{[(1R)-2,3-dihydro-1H-inden-1-yl]amino}quinolin-6-yl)-3-(propan-2-yl)urea

The compound is 5-HT5A receptor antagonist (Ki 2.5 nM).

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BRC0409
Product IDBRC0409
Product classBioreference compound
CAS number78246-49-8
MW365.8
Synonyms
BRL-29060A, FG-7051, Aropax, Brisdelle, Paxil, Pexeva, Sereupin, Seroxat,
Transport conditionsNormal

Paroxetine hydrochloride

Paroxetine, an antidepressant drug of the selective serotonin reuptake inhibitor (SSRI) type, has no active metabolites and has the highest specificity for serotonin receptors of all the SSRIs.

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BRC1017
Product IDBRC1017
Product classBioreference compound
CAS number316-07-4
MW371.3
Synonyms
Chlorpromazine sulfoxide hydrochloride; NSC 17470;
Transport conditionsNormal

Opromazine Hydrochloride

Opromazine hydrochloride is a derivative of Chlorpromazine, which is a dopamine antagonist of the typical antipsychotic class of medications possessing additional antiadrenergic, antiserotonergic, anticholinergic and antihistaminergic properties.

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BRC0730
Product IDBRC0730
Product classBioreference compound
CAS number52-86-8
MW375.9
Synonyms
MCN-JR-1625; NSC-170973; NSC-615296; R-1625; Dozic; Einalon S; Eukystol;
Transport conditionsNormal
Restrictions Included in California Proposition 65 list  WARNING! This product contains a chemical known to the State of California to cause health damage. For more information go to www.P65Warnings.ca.gov.

Haloperidol

Haloperidol is butyrophenone antipsychotic, D2, D3, and D4 dopamine receptor antagonist. It is used primarily to treat schizophrenia and other psychoses.

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BRC0605
Product IDBRC0605
Product classBioreference compound
CAS number863657-12-9
MW386.4
Synonyms
Transport conditionsNormal

N-[(2,6-dimethoxyphenyl)methyl]-N-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]guanidine

The compound is 5-HT5A antagonist.

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BRC0256
Product IDBRC0256
Product classBioreference compound
CAS number1098-60-8
MW388.9
Synonyms
Fluopromazine; Adazine; Psyquil;
Transport conditionsNormal

Triflupromazine hydrochloride

Triflupromazine hydrochloride binds to the dopamine D1 and dopamine D2 receptors and inhibits their activity.

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BRC0013
Product IDBRC0013
Product classBioreference compound
CAS number85650-56-2
MW401.8
Synonyms
Saphris,
Transport conditionsNormal

Asenapine maleate

Asenapine is a serotonin, dopamine, noradrenaline, and histamine antagonist in which asenapine possess more potent activity with serotonin receptors than dopamine. Asenapine is an atypical antipsychotic multireceptor neuroleptic drug which shows strong 5HT2A (serotonin) and D2 (dopamine) receptor antagonism, which has been shown to enhance dopamine (DA) and acetylcholine (Ach) efflux in rat brains. Asenapine may improve cognitive function and negative symptoms in patients with schizophrenia.

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BRC0397
Product IDBRC0397
Product classBioreference compound
CAS number130-61-0
MW407.0
Synonyms
Aldazine, Mallorol, Meleril, Mellaril, Mellerette, Melleretten, Melleril, Novoridazine, Ridazin, Ridazine, Sonapax, Thioril
Transport conditionsNormal

Thioridazine hydrochloride

Thioridazine is a trifluoro-methyl phenothiazine derivative intended for the management of schizophrenia and other psychotic disorders. It is a calcium channel protein inhibitor as well as a D2DR/D4DR inhibitor. It is an intercalating agent for analyzing the integrity of double stranded DNA by using the square-wave voltammetry.

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BRC0068
Product IDBRC0068
Product classBioreference compound
CAS number106266-06-2
MW410.5
Synonyms
Risperdal, Risperidal, Rispolept,
Transport conditionsNormal

Risperidone

Risperidone, a benzisoxazole derivative, is an atypical antipsychotic drug with high affinity for 5-hydrotryptamine (5-HT) and dopamine D2 receptors. It is used primarily in the management of schizophrenia, inappropriate behavior in severe dementia and manic episodes associated with bipolar I disorder.

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BRC0577
Product IDBRC0577
Product classBioreference compound
CAS number1809862-74-5
MW424.5
Synonyms
Transport conditionsNormal

3-methyloxetan-3-yl 4-[3-(2-methoxypyridin-3-yl)pyrazolo[1,5-a]pyrimidin-5-yl]piperazine-1-carboxylate

The compound is potent, brain penetrant inhibitor of AP2-associated protein kinase 1 (IC50 = 4.7 nM).

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BRC0084
Product IDBRC0084
Product classBioreference compound
CAS number129722-12-9
MW448.4
Synonyms
Abilify, Abilitat, Abilify Discmelt
Transport conditionsNormal

Aripiprazole

Aripiprazole is a psychotropic agent belonging to the chemical class of benzisoxazole derivatives and is indicated for the treatment of schizophrenia. Aripiprazole is a selective monoaminergic antagonist with high affinity for the serotonin Type 2 (5HT2), dopamine Type 2 (D2), 1 and 2 adrenergic, and H1 histaminergic receptors.

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BRC0517
Product IDBRC0517
Product classBioreference compound
CAS number866823-73-6
MW454.6
Synonyms
MRLSD 230, BINA
Transport conditionsNormal

Biphenylindanone A

Biphenyl-indanone A (BINA) is a potent selective positive allosteric modulator for the group II metabotropic glutamate receptor subtype mGluR2 (EC50 = 33.2 nM in CHO cells expressing human mGlu2). Exhibits antipsychotic and anxiolytic properties in mice.

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BRC0414
Product IDBRC0414
Product classBioreference compound
CAS number2062-78-4
MW461.6
Synonyms
NSC 170984, Orap, R 6238, Neoperidole, Opiran
Transport conditionsNormal
Restrictions Included in California Proposition 65 list  WARNING! This product contains a chemical known to the State of California to cause birth defects or other reproductive harm. For more information go to www.P65Warnings.ca.gov.

Pimozide

Pimozide is an orally active antipsychotic drug product which shares with other antipsychotics the ability to blockade dopaminergic receptors on neurons in the central nervous system.

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BRC0432
Product IDBRC0432
Product classBioreference compound
CAS number639089-54-6
MW464.6
Synonyms
VX-680, MK-0457
Transport conditionsNormal

Tozasertib

Tozasertib is a potent pan-ARK inhibitor but favors ARK-1 (Ki = 0.6 nM) over ARK-2 (Ki = 18 nM) or ARK-3 (Ki = 4.6 nM).

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BRC0025
Product IDBRC0025
Product classBioreference compound
CAS number440-17-5
MW480.4
Synonyms
Stelazine, Terfluzine, 440-17-5,
Transport conditionsNormal

Trifluoperazine dihydrochloride

Trifluoperazine is a trifluoro-methyl phenothiazine derivative intended for the management of schizophrenia and other psychotic disorders. Trifluoperazine has not been shown effective in the management of behaviorial complications in patients with mental retardation. Trifluoperazine blocks postsynaptic mesolimbic dopaminergic D1 and D2 receptors in the brain; depresses the release of hypothalamic and hypophyseal hormones and is believed to depress the reticular activating system thus affecting basal metabolism, body temperature, wakefulness, vasomotor tone, and emesis.

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BRC0402
Product IDBRC0402
Product classBioreference compound
CAS number84-02-6
MW606.1
Synonyms
Buccastem, Emetiral, Stemzine, Volimin
Transport conditionsNormal

Prochlorperazine dimaleate

Prochlorperazine is a piperazine phenothiazine related to high-potency neuroleptics such as perphenazine. It shares many of the actions and adverse effects of the antipsychotics.

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