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BRC0254
Product IDBRC0254
Product classBioreference compound
CAS number142-63-2
MW86.1
Synonyms
Diethylenediamine, Piperazidine, Piperazin, Antepar, Uvilon, Vermidol, Vermizine
Transport conditionsNormal

Piperazine Hexahydrate

Piperazine is a GABA receptor agonist.

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BRC1419
Product IDBRC1419
Product classBioreference compound
CAS number107-97-1
MW89.1
Synonyms
Methylglycine; N-Methylaminoacetic acid; Sarcosin; Sarcosinic acid;
Transport conditionsNormal

Sarcosine

Sarcosine is an endogenous inhibitor of GlyT1 with antipsychotic activity. It potentiates the action of glycine on the NMDA glycine binding site.

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BRC1147
Product IDBRC1147
Product classBioreference compound
CAS number22059-21-8
MW101.1
Synonyms
ACC; NSC 98430;
Transport conditionsNormal

ACPC

ACPC is NMDA receptor activity modulator, acts as a partial agonist at the glycine-binding site on NMDA receptors (EC50 = 0.7-0.9 µM) in the presence of low levels (1 µM) of glutamate and as a competitive antagonist at the glutamate-binding site on NMDA receptors (EC50 = 81.6 nM) with high levels (10 µM) of glutamate.

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BRC0928
Product IDBRC0928
Product classBioreference compound
CAS number68506-86-5
MW129.2
Synonyms
CPP-109; MDL 71,754; MDL-71754; RMI-71754; GVG; Sabril™; γ-Vinyl GABA;
Transport conditionsNormal

Vigabatrin

Vigabatrin is a structural analogue of gamma-aminobutyric acid, irreversible inhibitor of 4-aminobutyrate transaminase, the enzyme responsible for the catabolism of gamma-aminobutyric acid.

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BRC1068
Product IDBRC1068
Product classBioreference compound
CAS number3544-24-9
MW136.2
Synonyms
NSC 36962; SR 4294; WD 97-000835;
Transport conditionsNormal

INO-1001

INO-1001 is PARP (poly(ADP-ribose) polymerase) inhibitor (Ki = 1.8 μM), which protects cells from UV-B-induced apoptosis via influence on the cytoskeleton. Through its effects on PARPs, 3-amino benzamide causes telomere shortening and stimulates angiogenesis. It has PARP-mediated actions in such diverse diseases as atherosclerosis, neurogenesis, and cancer.

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BRC1029
Product IDBRC1029
Product classBioreference compound
CAS number59-50-7
MW142.6
Synonyms
NSC 4166; Neopredisan; Parol; Raschit; PCMC;
Transport conditionsNormal

Chlorocresol

Chlorocresol is a chlorinated phenol which is used as an antiseptic and preservative.

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BRC1362
Product IDBRC1362
Product classBioreference compound
CAS number19771-63-2
MW147.2
Synonyms
L-2-Oxo-4-thiazolidinecarboxylic acid; R-2-Oxo-1,3-thiazolidine-4-carboxylic acid;
Transport conditionsNormal

Procysteine

Procysteine is a precursor to glutathione (GSH) which is an important antioxidant. This compound has also been found to stimulate gene expression of insulin-like growth factor-1, cardiotrophin-1, and ciliary neurotrophic factor.

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BRC1023
Product IDBRC1023
Product classBioreference compound
CAS number700-06-1
MW147.2
Synonyms
NSC 525801; Indinol; I3C;
Transport conditionsNormal

Indole-3-carbinol

Indole-3-carbinol is a cell growth inhibitor that reversibly suppresses incorporation of [3H]thymidine in cells. It has been shown to have anti-cancer effects, at least in part through inhibition of NF-κB and Akt signaling pathways. Indole-3-carbinol displays the ability to inhibit endogenous retinoblastoma protein phosphorylation. Mechanistic studies suggest that in vitro this compound inhibits cell adhesion, migration, and invasion.

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BRC1035
Product IDBRC1035
Product classBioreference compound
CAS number41862-09-3
MW155.2
Synonyms
Transport conditionsNormal

6-Amino-1-ethyluracil

6-Amino-1-ethyluracil is A2B adenosine receptor antagonist, may used in prevention and treatment of liver disease.

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BRC1033
Product IDBRC1033
Product classBioreference compound
CAS number64-65-3
MW155.2
Synonyms
Mikedimide; NP 13; NSC 168667; NSC 58187; Zentraleptin;
Transport conditionsNormal

Bemegride

Bemegride is a central nervous system stimulant and antidote for barbiturate poisoning as its chemoreceptor agonism increases mean tidal volume, thereby increasing respiration and the concentration of O2 in blood.

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BRC1079
Product IDBRC1079
Product classBioreference compound
CAS number88-04-0
MW156.6
Synonyms
PCMX; Parametaxylenol; RBA 777;
Transport conditionsNormal

Chloroxylenol

Chloroxylenol is an antiseptic and disinfectant agent used for skin disinfection and cleaning surgical instruments.

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BRC0909
Product IDBRC0909
Product classBioreference compound
CAS number182485-36-5
MW161.1
Synonyms
Transport conditionsNormal

TPMPA

TPMPA is GABA receptor antagonist.

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BRC0818
Product IDBRC0818
Product classBioreference compound
CAS number616-91-1
MW163.2
Synonyms
5052; NSC-111180; RK-0202; NAC; Mercapturic acid;
Transport conditionsNormal

Acetylcysteine

Acetylcysteine (NAC) is an antioxidant and precursor of glutathione that has multiple effects in cells and animals. It is primarily used as a mucolytic agent and in the management of acetaminophen poisoning. It is essentially a prodrug that is converted to cysteine (in the intestine by the enzyme aminoacylase 1) and absorbed in the intestine into the bloodstream. As an antioxidant, NAC scavenges hydrogen peroxide, hydroxyl radical, and hypochlorous acid.

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BRC0692
Product IDBRC0692
Product classBioreference compound
CAS number76-38-0
MW165.0
Synonyms
DA-759; NSC-110432;
Transport conditionsNormal

Methoxyflurane

Methoxyflurane is an anesthetic used for induction and maintenance of general anesthesia. It induces muscle relaxation and reduces pains sensitivity by altering tissue excitability.

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BRC1066
Product IDBRC1066
Product classBioreference compound
CAS number498-02-2
MW166.2
Synonyms
NSC 209524; NSC 2146;
Transport conditionsNormal

Apocynin

Apocynin is a methoxy-substituted catechol that is commonly used as a selective NADPH-oxidase inhibitor with IC50 of 10 μM. Acts as an antioxidant in endothelial cells and vascular smooth muscle cells.

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BRC0189
Product IDBRC0189
Product classBioreference compound
CAS number60142-96-3
MW171.2
Synonyms
Gabapentin GR, Neurontin, Aclonium
Transport conditionsNormal

Gabapentin

Gabapentin interacts with cortical neurons at auxillary subunits of voltage-sensitive calcium channels. Gabapentin increases the synaptic concentration of GABA, enhances GABA responses at non-synaptic sites in neuronal tissues, and reduces the release of mono-amine neurotransmitters.

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BRC1392
Product IDBRC1392
Product classBioreference compound
CAS number57-08-9
MW173.2
Synonyms
NSC 12945; ε-Acetamidocaproic acid; CY 153; Acemin;
Transport conditionsNormal

Acexamic acid

Acexamic acid is related structurally to the antifibrinolytic agent aminocaproic acid. It is used for treatment of gastric ulcer or small bowel inflammation.

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BRC0615
Product IDBRC0615
Product classBioreference compound
CAS number2078-54-8
MW178.3
Synonyms
ICI 35868; Disoprivan; Disoprofol;
Transport conditionsNormal

Propofol

Propofol is a sedative-hypnotic agent for use in the induction and maintenance of anesthesia or sedation. It acts as a potentiator of the GABAA receptor.

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BRC0251
Product IDBRC0251
Product classBioreference compound
CAS number75448-53-2
MW180.2
Synonyms
Elixophyllin, Respbid, Theo-dur, Theolair, Uniphyl
Transport conditionsNormal

Theophylline

Theophylline, an xanthine derivative chemically similar to caffeine and theobromine, is used to treat asthma and bronchospasm. Theophylline has two distinct actions in the airways of patients with reversible (asthmatic) obstruction; smooth muscle relaxation (i.e., bronchodilation) and suppression of the response of the airways to stimuli (i.e., non-bronchodilator prophylactic effects).

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BRC0968
Product IDBRC0968
Product classBioreference compound
CAS number83-67-0
MW180.2
Synonyms
NSC-5039; SC-15090; Diurobromine;
Transport conditionsNormal

Theobromine

Theobromine is a purine alkaloid that is an adenosine receptor antagonist, weak PDE (phosphodiesterase) inhibitor. It is a diuretic and smooth-muscle relaxant.

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BRC0633
Product IDBRC0633
Product classBioreference compound
CAS number56-92-8
MW184.1
Synonyms
NSC-257873; NSC-33792;
Transport conditionsNormal

Histamine Dihydrochloride

Histamine is a depressor amine. It is a powerful stimulant of gastric secretion, a bronchoconstrictor, vasodilator, and also a centrally acting neurotransmitter.

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BRC0687
Product IDBRC0687
Product classBioreference compound
CAS number13838-16-9
MW184.5
Synonyms
Anesthetic 347; Alyrane;
Transport conditionsNormal

Enflurane

Enflurane is an anesthetic. It induces muscle relaxation and reduces pains sensitivity by altering tissue excitability. Enflurane acts as a positive allosteric modulator of the GABAA, glycine, and 5-HT3 receptors, and as a negative allosteric modulator of the AMPA, kainate, and NMDA receptors, as well as of nicotinic acetylcholine receptors.

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BRC0823
Product IDBRC0823
Product classBioreference compound
CAS number26675-46-7
MW184.5
Synonyms
R-E 235da1, HCFE 235da2,
Transport conditionsNormal

Isoflurane

Isoflurane is a general inhalation anesthetic. It induces a reduction in junctional conductance by decreasing gap junction channel opening times and increasing gap junction channel closing times.

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BRC0260
Product IDBRC0260
Product classBioreference compound
CAS number665-66-7
MW187.7
Synonyms
Aminoadamantane, Viregyt, Virosol, PK-Merz, Symadine, Symmetrel
Transport conditionsNormal
Restrictions Included in California Proposition 65 list Restriction  WARNING! This product contains a chemical known to the State of California to cause birth defects or other reproductive harm. For more information go to www.P65Warnings.ca.gov.

Amantadine hydrochloride

Amantadine is an antiviral drug which also acts as an antiparkinson agent, for which it is usually combined with L-DOPA when L-DOPA responses decline (probably due to tolerance).

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BRC0023
Product IDBRC0023
Product classBioreference compound
CAS number62-31-7
MW189.6
Synonyms
3-Hydroxytyramine, Deoxyepinephrine, Oxytyramine, Intropin, Revimine
Transport conditionsNormal

Dopamine hydrochloride

Dopamine is a natural catecholamine formed by the decarboxylation of 3,4-dihydroxyphenylalanine (DOPA). It is a precursor to norepinephrine in noradrenergic nerves and is also a neurotransmitter in certain areas of the central nervous system, especially in the nigrostriatal tract, and in a few peripheral sympathetic nerves. Dopamine produces positive chronotropic and inotropic effects on the myocardium, resulting in increased heart rate and cardiac contractility.

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BRC0295
Product IDBRC0295
Product classBioreference compound
CAS number58-08-2
MW194.2
Synonyms
Methyltheobromine, NSC 5036
Transport conditionsNormal

Caffeine

Central nervous system stimulant. Antagonist at A1 and A2A adenosine receptors and inhibitor of cyclic nucleotide phosphodiesterases. Mobilizes calcium from intracellular stores and inhibits benzodiazepine binding to GABA receptors.

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BRC0719
Product IDBRC0719
Product classBioreference compound
CAS number41078-02-8
MW194.2
Synonyms
3-Propylxanthine, D 4028
Transport conditionsNormal

Enprofylline

Enprofylline is a synthetic dimethylxanthine derivative, it antagonizes erythrocyte phosphodiesterase, increasing cAMP activity.

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BRC0595
Product IDBRC0595
Product classBioreference compound
CAS number67730-11-4
MW198.2
Synonyms
Transport conditionsNormal
Restrictions Included in California Proposition 65 list Restriction  WARNING! This product contains a chemical known to the State of California to cause cancer. For more information go to www.P65Warnings.ca.gov.

Glu-P1

Glu-P1 is an mutagenic compound.

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BRC1074
Product IDBRC1074
Product classBioreference compound
CAS number153322-05-5
MW198.3
Synonyms
ARL 15896; FPL 15896; AR-R15896; AZD6765;
Transport conditionsNormal

Lanicemine

Lanicemine is a non-selective, voltage-dependent NMDA channel blocker (IC50 = 4-7 µM). It has been used in trials studying the treatment and basic science of Depression, Major Depressive Disorder, and Treatment-Resistant Major Depressive Disorder.

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BRC0390
Product IDBRC0390
Product classBioreference compound
CAS number55-65-2
MW198.3
Synonyms
Ismedine, Ismelin
Transport conditionsNormal

Guanethidine

Guanethidine works by decreasing the heart rate and relaxing the blood vessels so that blood can flow more easily through the body, thereby reducing these risks. It is a postganglionic sympathetic nerve terminal blocker that prevents the release of norepinephrine from nerve terminals.

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BRC0550
Product IDBRC0550
Product classBioreference compound
CAS number19772-76-0
MW199.2
Synonyms
DL-Willardiine
Transport conditionsNormal

(±)-Willardiine

(±)-Willardiine is a selective inhibitor of specific binding of [3H]AMPA to Ionotropic glutamate receptor AMPA (IC50 = 1800 nM).

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BRC0857
Product IDBRC0857
Product classBioreference compound
CAS number28523-86-6
MW200.1
Synonyms
Transport conditionsNormal

Sevoflurane

Sevoflurane is one of the most commonly used volatile anesthetic agents, particularly for outpatient anesthesia, across all ages, as well as in veterinary medicine.

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BRC0637
Product IDBRC0637
Product classBioreference compound
CAS number2809-21-4
MW206.0
Synonyms
M05BA01; NSC-227995; EHDP; HEDP; Hydroxyethylidene Diphosphonic Acid;
Transport conditionsNormal

Etidronic acid

Etidronate is a first generation, non-nitrogenous diphosphonate analog of endogenous pyrophosphate. It affects on calcium metabolism, inhibits ectopic calcification and slows down bone resorption and bone turnover.

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BRC0150
Product IDBRC0150
Product classBioreference compound
CAS number1313437-84-1
MW209.9
Synonyms
Trilithium citrate
Transport conditionsNormal
Restrictions Included in California Proposition 65 list Restriction  WARNING! This product contains a chemical known to the State of California to cause health damage. For more information go to www.P65Warnings.ca.gov.

Lithium Citrate

Lithium salts such as lithium carbonate, lithium citrate, and lithium orotate are mood stabilizers. They are used in the treatment of bipolar disorder, since unlike most other mood altering drugs, they counteract both mania and depression.

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BRC1008
Product IDBRC1008
Product classBioreference compound
CAS number55206-24-1
MW214.7
Synonyms
Transport conditionsNormal

6-fluorotryptamine hydrochloride

6-fluorotryptamine hydrochloride is a tryptamine derivative that potentially agonizes 5-HT serotonin receptors (EC50 = 4.56 nM).

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BRC0032
Product IDBRC0032
Product classBioreference compound
CAS number41100-52-1
MW215.8
Synonyms
Abixa, Akatinol, Axura, Memox
Transport conditionsNormal

Memantine hydrochloride

Memantine exerts its action through uncompetitive NMDA receptor antagonism, binding preferentially to the NMDA receptor-operated cation channels. Memantine also has antagonistic activity at the type 3 serotonergic (5-HT3) receptor with a potency that is similar to that at the NMDA receptor, and lower antagonistic activity at the nicotinic acetylcholine receptor. This drug has no affinity for γ-aminobutyric acid (GABA), benzodiazepine, dopamine, adrenergic, histamine, or glycine receptors or for voltage-dependent calcium, sodium, or potassium channels.

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BRC0226
Product IDBRC0226
Product classBioreference compound
CAS number125-33-7
MW218.3
Synonyms
Desoxyphenobarbital, Mysoline, Liskantin, Mizodin, Mylepsinum, Pridona, Primid, Prysoline, Sertan
Transport conditionsNormal
Restrictions Included in DEA controlled list Restriction

Primidone

An antiepileptic agent related to the barbiturates; it is partly metabolized to phenobarbital in the body and owes some of its actions to this metabolite. Primidone is a GABA receptor agonist.

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BRC0180
Product IDBRC0180
Product classBioreference compound
CAS number364-98-7
MW230.7
Synonyms
Eudemine, Hyperstat, Sch-6783, SRG-95213, Proglycem
Transport conditionsNormal

Diazoxide

Diazoxide is a potassium channel activator, which causes local relaxation in smooth muscle by increasing membrane permeability to potassium ions. This switches off voltage-gated calcium ion channels which inhibits the generation of an action potential.

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BRC0052
Product IDBRC0052
Product classBioreference compound
CAS number1744-22-5
MW234.2
Synonyms
Rilutek, RP-54274, PK 26124
Transport conditionsNormal

Riluzole

Psychotropic agent with anticonvulsant, hypnotic, anxiolytic, anti-ischemic and anesthetic properties. Inhibits glutamate release from presynaptic terminals and increases Na+-dependent glutamate uptake in rat cortical synaptosomes. Blocks voltage-dependent Na+ channels and inhibits GABA uptake by striatal synaptosomes; neuroprotective.

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BRC0239
Product IDBRC0239
Product classBioreference compound
CAS number25451-15-4
MW238.2
Synonyms
Taloxa, ADD-03055
Transport conditionsNormal

Felbamate

Felbamate is an anticonvulsant drug used in the treatment of epilepsy. It has a weak inhibitory effect on GABA receptor binding sites.

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BRC1086
Product IDBRC1086
Product classBioreference compound
CAS number1955540-15-4
MW239.7
Synonyms
Transport conditionsNormal

3-phenoxy-8-azabicyclo[3.2.1]octane hydrochloride

3-phenoxy-8-azabicyclo[3.2.1]octane hydrochloride is inhibitor of [3H]noradrenaline, [3H]dopamine and [3H]serotonin reuptake.

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BRC0178
Product IDBRC0178
Product classBioreference compound
CAS number36791-04-5
MW244.2
Synonyms
RBV; Rebretron; Ribamide; Vilona; Viramid; Virazide; NSC-163039; ICN-1229; RTCA; Tribavirin;
Transport conditionsNormal
Restrictions Included in California Proposition 65 list Restriction  WARNING! This product contains a chemical known to the State of California to cause birth defects or other reproductive harm. For more information go to www.P65Warnings.ca.gov.

Ribavirin

Ribavirin is a guanosine analog with antiviral properties against DNA and RNA viruses, including respiratory syncytial virus, hepatitis C, and influenza.

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BRC0445
Product IDBRC0445
Product classBioreference compound
CAS number33125-97-2
MW244.3
Synonyms
Lipuro, Propiscin, R 16659, Hypnomidate, Amidate
Transport conditionsNormal

Etomidate

Etomidate is an imidazole compound that appears to depress CNS function via GABA and categorized as an anesthetic. Etomidate also inhibits adrenal cortisol biosynthesis and mitigates hypercortisolism, as is found in Cushing syndrome.

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BRC1061
Product IDBRC1061
Product classBioreference compound
CAS number77191-36-7
MW246.3
Synonyms
DM 9384; DMMPA; DMPPA; DZL 221; Translon;
Transport conditionsNormal

Nefiracetam

Nefiracetam is cognitive enhancer that displays various pharmacological effects. Activates L/N-type calcium channels, cholinergic, monoaminergic and GABAergic systems. Displays potent neuroprotective action in the retinal ischemia-reperfusion model in vivo.

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BRC0973
Product IDBRC0973
Product classBioreference compound
CAS number66376-36-1
MW249.1
Synonyms
G 704650; GTH 4; L 670; L 670452; MK 217; ABDP;
Transport conditionsNormal

Alendronic acid

Alendronate is a second-generation bisphosphonate. Used to reduce hypercalcemia in tumor-induced bone disease, to treat corticosteroid-induced osteoporosis and Pagets disease.

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BRC0246
Product IDBRC0246
Product classBioreference compound
CAS number28311-31-1
MW250.1
Synonyms
(+-)-Baclofen, Baclon, Kemstro, Lioresal Intrathecal,
Transport conditionsNormal

Baclofen hydrochloride

Baclofen is a direct agonist at GABAB receptors.

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BRC0464
Product IDBRC0464
Product classBioreference compound
CAS number4815-38-7
MW261.3
Synonyms
Transport conditionsNormal

Ethyl 2-Amino-4-methyl-5-phenylthiophene-3-carboxylate

Glutamate receptors inhibitor.

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BRC0421
Product IDBRC0421
Product classBioreference compound
CAS number85650-52-8
MW265.4
Synonyms
Org 3770, 6-Azamianserin, Avanza, Axit, Mirtabene, Mirtaz, Mirtazon, Norset, Promyrtil, Remergil, Remergon, Remeron, Remeron SolTab, Rexer, Zispin
Transport conditionsNormal

Mirtazapine

Mirtazapine, an antidepressant of the piperazinoazepine class, is a tetracyclic compound with an anxiolytic effect. Mirtazapine has fewer ADRs than tricyclic antidepressants and is better tolerated. Selective blockade of specific serotonin receptors by mirtazapine likey minimizes side effects typical of other antidepressants.

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BRC0828
Product IDBRC0828
Product classBioreference compound
CAS number58-61-7
MW267.2
Synonyms
SR-96225; USAF CB-10; Ado;
Transport conditionsNormal

Adenosine

Adenosine is an endogenous nucleoside. It activates purine receptors, as well as relax vascular smooth muscles through the reduction in calcium uptake by inhibition of slow inward calcium current and activation of adenylate cyclase in smooth muscle cells.

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BRC0138
Product IDBRC0138
Product classBioreference compound
CAS number53910-25-1
MW268.3
Synonyms
Deoxycoformycin; Nipent; 2-Deoxycoformycin;
Transport conditionsNormal
Restrictions Included in California Proposition 65 list Restriction  WARNING! This product contains a chemical known to the State of California to cause birth defects or other reproductive harm. For more information go to www.P65Warnings.ca.gov.

Pentostatin

Pentostatin is a potent transition state inhibitor of adenosine deaminase (ADA), the greatest activity of which is found in cells of the lymphoid system.

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