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Androgen receptor

StructureProduct infoAvailabilityQuantity / Price
BRC0993
Product IDBRC0993
Product classBioreference compound
CAS number65-45-2
MW137.1
Synonyms
OHB;
Transport conditionsNormal

Salicylamide

Salicylamide is an analgesic and antipyretic agent. Its medicinal uses are similar to those of aspirin.

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BRC0969
Product IDBRC0969
Product classBioreference compound
CAS number97-53-0
MW164.2
Synonyms
NSC-209525; NSC-8895; 4-allylguaiacol;
Transport conditionsNormal

Eugenol

Eugenol is an antifungal and antimicrobial agent, TRPV1 receptor agonist. Its exact mechanism of action is unknown, however, it has been shown to interfere with action potential conduction.

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BRC1071
Product IDBRC1071
Product classBioreference compound
CAS number120-47-8
MW166.2
Synonyms
Mycocten; NSC 23514; NSC 8510; E 214; Easeptol;
Transport conditionsNormal

Ethylparaben

Ethylparaben is the ethyl ester of p-hydroxybenzoic acid, used as an anti-microbial agent and food additive. It is a standardized chemical allergen. The physiologic effect of ethylparaben is by means of increased histamine release, and cell-mediated immunity.

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BRC1080
Product IDBRC1080
Product classBioreference compound
CAS number94-25-7
MW193.2
Synonyms
Butylcaine; Hemoride; NSC 128464; Planoform; Scuroform;
Transport conditionsNormal

Butamben

Butamben is a mildly water-soluble, long-duration local anesthetic that is thought to reversibly blocking nerve conduction.

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BRC1077
Product IDBRC1077
Product classBioreference compound
CAS number94-26-8
MW194.2
Synonyms
NSC 13164; NSC 8475; Nipabutyl; SPF;
Transport conditionsNormal

Butylparaben

Butylparaben is an antifungal preservative in cosmetic products.

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BRC0858
Product IDBRC0858
Product classBioreference compound
CAS number131-57-7
MW228.2
Synonyms
NSC-7778; Benzophenone-3;
Transport conditionsNormal

Oxybenzone

Oxybenzone is a derivative of benzophenone. It is used as an ingredient in sunscreen and other cosmetics because it absorbs UV-A ultraviolet rays.

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BRC0684
Product IDBRC0684
Product classBioreference compound
CAS number56-53-1
MW268.4
Synonyms
NSC 3070, DES
Transport conditionsNormal
Restrictions Included in California Proposition 65 list  WARNING! This product contains a chemical known to the State of California to cause cancer and birth defects or other reproductive harm. For more information go to www.P65Warnings.ca.gov.

Diethylstilbestrol

Diethylstilbestrol is a synthetic estrogen with carcinogenic properties (estrogen receptor agonist, EC50 = 0.007 nM). Used in the treatment of prostate cancer to block the production of testosterone.

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BRC0796
Product IDBRC0796
Product classBioreference compound
CAS number53-16-7
MW270.4
Synonyms
NSC 9699, WAY 164397
Transport conditionsNormal
Restrictions Included in California Proposition 65 list  WARNING! This product contains a chemical known to the State of California to cause cancer. For more information go to www.P65Warnings.ca.gov.

Estrone

Estrone is an estradiol metabolite, estrogen receptor agonist.

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BRC0142
Product IDBRC0142
Product classBioreference compound
CAS number13311-84-7
MW276.2
Synonyms
Eulexin, Niftolide, Drogenil, SCH-13521
Transport conditionsNormal
Restrictions Included in California Proposition 65 list  WARNING! This product contains a chemical known to the State of California to cause birth defects or other reproductive harm. For more information go to www.P65Warnings.ca.gov.

Flutamide

Flutamide is a nonsteroidal antiandrogen that blocks the action of both endogenous and exogenous testosterone by binding to the androgen receptor. In addition Flutamide is a potent inhibitor of testosterone-stimulated prostatic DNA synthesis. Moreover, it is capable of inhibiting prostatic nuclear uptake of androgen.

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BRC0479
Product IDBRC0479
Product classBioreference compound
CAS number530-78-9
MW281.2
Synonyms
Arlef, CI 440, CN 27544, INF 1837, NSC 219007, NSC 82699
Transport conditionsNormal

Flufenamic acid

Flufenamic acid is an anthranilic acid-derived nonsteroidal anti-inflammatory drug (NSAID) thought to exert its actions by a prostanoid-independent mechanism.

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BRC0136
Product IDBRC0136
Product classBioreference compound
CAS number52806-53-8
MW292.2
Synonyms
Hydroxyniphtholide, Sch 16423
Transport conditionsNormal

Hydroxyflutamide

2-hydroxy Flutamide is the major metabolite formed during the metabolism of the non-steroidal antiandrogen flutamide by cytochrome P450 (CYP) isoforms CYP1A2 and CYP3A4. Through competitive inhibition of the binding of testosterone to the nuclear androgen receptor (AR; IC50 = ~ 300-900), 2-hydroxy flutamide blocks the expression of AR target genes and prevents androgen-dependent stabilization of the AR.

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BRC0043
Product IDBRC0043
Product classBioreference compound
CAS number797-63-7
MW312.5
Synonyms
Levonorgestrel, Methylnorethindrone, Logynon, Nordette, Eugynon, Microgynon, Ovran, Ovranette, Trinordiol
Transport conditionsNormal
Restrictions Included in DEA controlled list

(-) - Norgestrel

(-) - Norgestrel is a synthetic progesterone analog and the biologically active component of norgestrel, which is a racemic mixture. Levonorgestrel prevents pregnancy by inhibiting ovulation and by causing the cervical mucous to thicken, which makes it harder for sperm to move toward the uterus. Levonorgestrel exhibits approximately three-times higher binding affinity than progesterone for the progesterone receptor.

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BRC0866
Product IDBRC0866
Product classBioreference compound
CAS number57-83-0
MW314.5
Synonyms
BP 14, NSC-64377, NSC-9704, U 3672
Transport conditionsNormal
Restrictions Included in California Proposition 65 list  WARNING! This product contains a chemical known to the State of California to cause health damage. For more information go to www.P65Warnings.ca.gov.

Progesterone

Progesterone is steroid hormone produced by the corpus luteum. It is endogenous progesterone receptor (PR) agonist (EC50 = 0.5 nM).

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BRC0940
Product IDBRC0940
Product classBioreference compound
CAS number63612-50-0
MW317.2
Synonyms
RU-23908;
Transport conditionsNormal

Nilutamide

Nilutamide is an antineoplastic hormonal agent, nonsteroidal anti-androgen with selectivity for androgen receptors.

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BRC0339
Product IDBRC0339
Product classBioreference compound
CAS number66778-17-4
MW340.3
Synonyms
Aesculin
Transport conditionsNormal

Esculin

The main activities of Esculine focus on capillary protection, as it improves capillary permeability and fragility. It is reported to inhibit catabolic enzymes such as hyaluronidase and collagenase, thus preserving the integrity of the perivascular connective tissue.

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BRC0048
Product IDBRC0048
Product classBioreference compound
CAS number976-71-6
MW340.5
Synonyms
Phanurane, Aldadiene, Luvion, Aldadiene,
Transport conditionsNormal

Canrenone

Mineralocorticoid receptor antagonist. Active metabolite of spironolactone. A potassium sparing diuretic that acts by antagonism of aldosterone in the distal renal tubules. It is used mainly in the treatment of refractory edema in patients with congestive heart failure, nephrotic syndrome, or hepatic cirrhosis. Its effects on the endocrine system are utilized in the treatments of hirsutism and acne but they can lead to adverse effects.

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BRC1281
Product IDBRC1281
Product classBioreference compound
CAS number335-67-1
MW414.1
Synonyms
A 5717; EF 201; Eftop EF 201; NSC 95114; PFOA;
Transport conditionsNormal
Restrictions Included in California Proposition 65 list  WARNING! This product contains a chemical known to the State of California to cause health damage. For more information go to www.P65Warnings.ca.gov.

Perfluorooctanoic acid

Perfluorooctanoic acid is one of the most commonly used perfluorinated compounds, it causes hepatic peroxisome proliferation in rodents. It may have toxic effects on the immune system, liver, development, and endocrine systems through alteration of DNA methylation enzymes.

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BRC0072
Product IDBRC0072
Product classBioreference compound
CAS number52-01-7
MW416.6
Synonyms
Aldactone, Verospiron, Spiroctan
Transport conditionsNormal
Restrictions Included in California Proposition 65 list  WARNING! This product contains a chemical known to the State of California to cause cancer. For more information go to www.P65Warnings.ca.gov.

Spironolactone

Spironolactone is a potent antagonist of the androgen receptor with IC50 of 77 nM. Spironolactone is a synthetic 17-lactone steroid which is a renal competitive aldosterone antagonist in a class of pharmaceuticals called potassium-sparing diuretics.

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BRC0027
Product IDBRC0027
Product classBioreference compound
CAS number126784-99-4
MW475.6
Synonyms
EllaOne, Ella, CDB 2914,
Transport conditionsNormal

Ulipristal acetate

Ulipristal is a selective, reversible progestin receptor modulator and its tissue targets include the uterus, cervix, ovaries, and hypothalamus. Ulipristal may act as an agonist or antagonist in the presence or absence of progesterone based on the tissue target.

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BRC0646
Product IDBRC0646
Product classBioreference compound
CAS number146-56-5
MW510.4
Synonyms
SQ 10733, Squibb 16144, Moditen, OMCA, Anatensol, Trancin, Valamina
Transport conditionsNormal

Fluphenazine dihydrochloride

Fluphenazine dihydrochloride is a phenothiazine-class D1DR and D2DR inhibitor. Intended for the management of schizophrenia and other psychotic disorders.

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BRC0901
Product IDBRC0901
Product classBioreference compound
CAS number65277-42-1
MW531.4
Synonyms
Phytorol, R 41400, Tocon
Transport conditionsNormal

Ketoconazole

Ketoconazole is anti-fungal agent with potent anti-metastatic, anti-neoplastic, and anti-psoriatic activities. It is an inhibitor of cytochrome P-450 in steroid biosynthesis. Also acts as an inhibitor of 5-lipoxygenase and thromboxane synthase activities.

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