EnamineStore

Welcome, Guest
Tutorials

Analgesics

StructureProduct infoAvailabilityQuantity / Price
BRC0993
Product IDBRC0993
Product classBioreference compound
CAS number65-45-2
MW137.1
Synonyms
OHB;
Transport conditionsNormal

Salicylamide

Salicylamide is an analgesic and antipyretic agent. Its medicinal uses are similar to those of aspirin.

Product Page

In Stock(5 business days)  
BRC0859
Product IDBRC0859
Product classBioreference compound
CAS number69-72-7
MW138.1
Synonyms
FEMA NO. 3985; K-557; NSC-180;
Transport conditionsNormal

Salicylic acid

Salicylic acid is bacteriostatic, fungicide and keratolytic agent. It is directly and irreversibly inhibits the activity of COX-1 and COX-2 to decrease the formation of precursors of prostaglandins and thromboxanes from arachidonic acid.

Product Page

In Stock(5 business days)  
BRC0873
Product IDBRC0873
Product classBioreference compound
CAS number67-48-1
MW139.6
Synonyms
Bilineurine;
Transport conditionsNormal

Choline

Choline is a precursor to acetylcholine. It is needed for good nerve conduction throughout the CNS. Choline is also needed for gallbladder regulation, liver function, and lecithin formation; for cholesterol metabolism and prevents excessive fat build up in the liver.

Product Page

In Stock(5 business days)  
BRC0981
Product IDBRC0981
Product classBioreference compound
CAS number103-90-2
MW151.2
Synonyms
NSC-109028; NSC-3991; APAP; Acenol; Paracetamol;
Transport conditionsNormal

Acetaminophen

Acetaminophen is a widely used analgesic and antipyretic drug that is used for the relief of fever, headaches, and other minor aches and pains. It is thought to act primarily in the CNS, increasing the pain threshold by inhibiting both isoforms of cyclooxygenase, COX-1, COX-2, and COX-3 enzymes involved in prostaglandin synthesis.

Product Page

In Stock(5 business days)  
BRC0168
Product IDBRC0168
Product classBioreference compound
CAS number89-57-6
MW153.1
Synonyms
5-ASA, Asacol, Asacolitin, Canasa, Claversal, Fisalamine, Iialda, Lixacol, m-Aminosalicylic acid, P-Aminosalicylsaeure, Pentasa, Rowasa, Salofalk
Transport conditionsNormal

Mesalazine

An anti-inflammatory agent, structurally related to the salicylates, which is active in inflammatory bowel disease. It is considered to be the active moiety of sulphasalazine. 

Product Page

In Stock(5 business days)  
BRC1290
Product IDBRC1290
Product classBioreference compound
CAS number97-59-6
MW158.1
Synonyms
NSC 7606; Psoralon; SD 101; Sebical;
Transport conditionsNormal

Allantoin

Allantoin is a purine metabolite via the uric acid pathway. It may be a useful biomarker for oxidative stress.

Product Page

In Stock(5 business days)  
BRC0692
Product IDBRC0692
Product classBioreference compound
CAS number76-38-0
MW165.0
Synonyms
DA-759; NSC-110432;
Transport conditionsNormal

Methoxyflurane

Methoxyflurane is an anesthetic used for induction and maintenance of general anesthesia. It induces muscle relaxation and reduces pains sensitivity by altering tissue excitability.

Product Page

In Stock(5 business days)  
BRC1066
Product IDBRC1066
Product classBioreference compound
CAS number498-02-2
MW166.2
Synonyms
NSC 209524; NSC 2146;
Transport conditionsNormal

Apocynin

Apocynin is a methoxy-substituted catechol that is commonly used as a selective NADPH-oxidase inhibitor with IC50 of 10 μM. Acts as an antioxidant in endothelial cells and vascular smooth muscle cells.

Product Page

In Stock(5 business days)  
BRC1078
Product IDBRC1078
Product classBioreference compound
CAS number149-91-7
MW170.1
Synonyms
NSC 20103; NSC 674319;
Transport conditionsNormal

Gallic acid

Gallic acid is an anti-inflammatory agent and cyclooxygenase inhibitor found in plants and has been shown to Induce apoptosis in human lung cancer cells. It is often used as a standard for determining the phenol content of various analytes by the Folin-Ciocalteau assay where results are reported in gallic acid equivalents.

Product Page

In Stock(5 business days)  
BRC0189
Product IDBRC0189
Product classBioreference compound
CAS number60142-96-3
MW171.2
Synonyms
Gabapentin GR, Neurontin, Aclonium
Transport conditionsNormal

Gabapentin

Gabapentin interacts with cortical neurons at auxillary subunits of voltage-sensitive calcium channels. Gabapentin increases the synaptic concentration of GABA, enhances GABA responses at non-synaptic sites in neuronal tissues, and reduces the release of mono-amine neurotransmitters.

Product Page

In Stock(5 business days)  
BRC0319
Product IDBRC0319
Product classBioreference compound
CAS number62-44-2
MW179.2
Synonyms
Achrocidin, Codempiral, Commotional, Contradol, Contradouleur
Transport conditionsNormal
Restrictions Included in California Proposition 65 list  WARNING! This product contains a chemical known to the State of California to cause cancer. For more information go to www.P65Warnings.ca.gov.

Phenacetin

Phenacetin was the first NSAID and fever reducer to go on the market. Its analgesic effects are due to its actions on the sensory tracts of the spinal cord. In addition, phenacetin has a depressant action of the heart, where it acts as a negative inotrope.

Product Page

In Stock(5 business days)  
BRC0936
Product IDBRC0936
Product classBioreference compound
CAS number50-78-2
MW180.2
Synonyms
BAY1019036; NSC-27223; NSC-406186; ASA; Aspirin;
Transport conditionsNormal
Restrictions Included in California Proposition 65 list  WARNING! This product contains a chemical known to the State of California to cause birth defects or other reproductive harm. For more information go to www.P65Warnings.ca.gov.

Acetylsalicylic acid

Acetylsalicylic acid is an anti-inflammatory and antipyretic agent and acts as the inhibitor of cyclooxygenase which results in the inhibition of the biosynthesis of prostaglandins. It also inhibits platelet aggregation and is used in the prevention of arterial and venous thrombosis.

Product Page

In Stock(5 business days)  
BRC0260
Product IDBRC0260
Product classBioreference compound
CAS number665-66-7
MW187.7
Synonyms
Aminoadamantane, Viregyt, Virosol, PK-Merz, Symadine, Symmetrel
Transport conditionsNormal
Restrictions Included in California Proposition 65 list  WARNING! This product contains a chemical known to the State of California to cause birth defects or other reproductive harm. For more information go to www.P65Warnings.ca.gov.

Amantadine hydrochloride

Amantadine is an antiviral drug which also acts as an antiparkinson agent, for which it is usually combined with L-DOPA when L-DOPA responses decline (probably due to tolerance).

Product Page

In Stock(5 business days)  
BRC0978
Product IDBRC0978
Product classBioreference compound
CAS number60-80-0
MW188.2
Synonyms
Transport conditionsNormal

Antipyrine

Antipyrine is an analgesic and antipyretic. It inhibits isoforms of cyclooxygenase, COX-1, COX-2, and COX-3 enzymes involved in prostaglandin (PG) synthesis. Antipyrine is often used in testing the effects of other drugs or diseases on drug-metabolizing enzymes in the liver.

Product Page

In Stock(5 business days)  
BRC0827
Product IDBRC0827
Product classBioreference compound
CAS number51146-56-6
MW206.3
Synonyms
d-ibuproten; S(+)-ibuprofen;
Transport conditionsNormal

Dexibuprofen

Dexibuprofen is a non-steroidal anti-inflammatory drug. It is a pharmacologically effective enantiomer of racemic ibuprofen that differs in physicochemical properties.

Product Page

In Stock(5 business days)  
BRC0814
Product IDBRC0814
Product classBioreference compound
CAS number15687-27-1
MW206.3
Synonyms
NSC 256857; U-18753;
Transport conditionsNormal

Ibuprofen

Ibuprofen is a nonsteroidal anti-inflammatory agent with analgesic and antipyretic properties. It is a non-selective, reversible COX inhibitor (IC50 for human recombinant COX-1 and COX-2 are 2.6 and 1.53 µM, respectively).

Product Page

In Stock(5 business days)  
BRC0308
Product IDBRC0308
Product classBioreference compound
CAS number7361-61-7
MW220.3
Synonyms
Anased, ROMPUN, Solvazine, Gemini, Chanazine, Bayer 1470, Tranquived, Xyla-Ject
Transport conditionsNormal

Xylazine

Xylazine is a potent α2 adrenergic agonist. Due to xylazine’s highly lipophilic nature, xylazine directly stimulates central α2 receptors as well as peripheral α-adrenoceptors in a variety of tissues.

Product Page

In Stock(5 business days)  
BRC0826
Product IDBRC0826
Product classBioreference compound
CAS number22204-53-1
MW230.3
Synonyms
RS-3540;
Transport conditionsNormal

Naproxen

Naproxen is a member of the arylacetic acid group of nonsteroidal anti-inflammatory drugs with analgesic and antipyretic properties. It is non-selective cyclooxygenase inhibitor. Has a neuroprotective role against colchicine-induced cognitive impairment and oxidative stress.

Product Page

In Stock(5 business days)  
BRC0926
Product IDBRC0926
Product classBioreference compound
CAS number298-46-4
MW236.3
Synonyms
G-32883; GEIGY 32883; NSC-169864; SPD417; CBZ;
Transport conditionsNormal
Restrictions Included in California Proposition 65 list  WARNING! This product contains a chemical known to the State of California to cause birth defects or other reproductive harm. For more information go to www.P65Warnings.ca.gov.

Carbamazepine

Carbamazepine is an anticonvulsant used to control grand mal and psychomotor or focal seizures. It inhibits neuronal voltage-gated Na+ channels. Potentiates GABA-induced Cl- currents in HEK 293 cells expressing the GABAA receptor α1β2γ2 subtype combination. Can induce autophagy by inhibiting inositol synthesis.

Product Page

In Stock(5 business days)  
BRC0187
Product IDBRC0187
Product classBioreference compound
CAS number111406-87-2
MW236.3
Synonyms
Zyflo, ICI D2138
Transport conditionsNormal
Restrictions Included in California Proposition 65 list  WARNING! This product contains a chemical known to the State of California to cause cancer and birth defects or other reproductive harm. For more information go to www.P65Warnings.ca.gov.

Zileuton

Zileuton is an asthma drug that differs chemically and pharmacologically from other antiasthmatic agents. It blocks leukotriene synthesis by inhibiting 5-lipoxygenase, an enzyme of the eicosanoid synthesis pathway.

Product Page

In Stock(5 business days)  
BRC0004
Product IDBRC0004
Product classBioreference compound
CAS number145108-58-3
MW236.7
Synonyms
Precedex, Dex, Dexmedetomidine HCL, (S)-Medetomidine hydrochloride
Transport conditionsNormal

Dexmedetomidine hydrochloride

Dexmedetomidine (hydrochloride) is the (S)-enantiomer of medetomidine (racemic form of this compound), a highly selective, potent and specific agonist of 2-adrenergic receptor (2-adrenoceptor).

Product Page

In Stock(5 business days)  
BRC0971
Product IDBRC0971
Product classBioreference compound
CAS number61-68-7
MW241.3
Synonyms
CI-473; CN-35355; INF-3355; J2.344B; M01AG01;
Transport conditionsNormal

Mefenamic acid

Mefenamic acid is a member of the fenamate group of nonsteroidal anti-inflammatory drugs. It exhibits anti-inflammatory, analgesic, and antipyretic activities. Mefenamic acid is a noncompetitive inhibitor of 2-arachidonoylglycerol oxygenation and a competitive inhibitor of COX-2 oxygenation of arachidonic acid.

Product Page

In Stock(5 business days)  
BRC1004
Product IDBRC1004
Product classBioreference compound
CAS number36330-85-5
MW254.3
Synonyms
CL 82,204;
Transport conditionsNormal

Fenbufen

Fenbufen is a non-steroidal anti-inflammatory drug. Used primarily to treat inflammation in osteoarthritis, ankylosing spondylitis, and tendinitis. It can also be used to relieve backaches, sprains, and fractures.

Product Page

In Stock(5 business days)  
BRC0718
Product IDBRC0718
Product classBioreference compound
CAS number22071-15-4
MW254.3
Synonyms
Orudis; Oruvail;
Transport conditionsNormal

Ketoprofen

Ketoprofen is a nonsteroidal anti-inflammatory agent with analgesic and antipyretic properties. It is used to treat rheumatoid arthritis, osteoarthritis, dysmenorrhea, and alleviate moderate pain. Ketoprofen is a non-selective NSAID exhibiting IC50 values of 0.5 µM and 2.33 µM for human recombinant COX-1 and COX-2, respectively.

Product Page

In Stock(5 business days)  
BRC0413
Product IDBRC0413
Product classBioreference compound
CAS number74103-06-3
MW255.3
Synonyms
Acular LS®, Acular PF®, RS 37619, Sprix®, Bedoral, Dolten,
Transport conditionsNormal

Ketorolac

Ketorolac is a nonsteroidal anti-inflammatory drug (NSAID) chemically related to indomethacin and tolmetin. Ketorolac tromethamine is a racemic mixture of [-]S- and [+]R-enantiomeric forms, with the S-form having analgesic activity.

Product Page

In Stock(5 business days)  
BRC0889
Product IDBRC0889
Product classBioreference compound
CAS number4205-91-8
MW266.6
Synonyms
ST 155, ST 155-BS
Transport conditionsNormal

Clonidine hydrochloride

Clonidine is an hypotensive agent, centrally-acting α2-adrenergic agonist.

Product Page

In Stock(5 business days)  
BRC0828
Product IDBRC0828
Product classBioreference compound
CAS number58-61-7
MW267.2
Synonyms
SR-96225; USAF CB-10; Ado;
Transport conditionsNormal

Adenosine

Adenosine is an endogenous nucleoside. It activates purine receptors, as well as relax vascular smooth muscles through the reduction in calcium uptake by inhibition of slow inward calcium current and activation of adenylate cyclase in smooth muscle cells.

Product Page

In Stock(5 business days)  
BRC1295
Product IDBRC1295
Product classBioreference compound
CAS number51298-62-5
MW269.7
Synonyms
Transport conditionsNormal

L-NAME hydrochloride

L-NAME hydrochloride is a nonselective inhibitor of nitric oxide synthetases.

Product Page

In Stock(5 business days)  
BRC0203
Product IDBRC0203
Product classBioreference compound
CAS number108605-62-5
MW270.2
Synonyms
a 77-1726; Aubagio; HMR1726;
Transport conditionsNormal

(E, Z) - Teriflunomide

Teriflunomide is an immunomodulatory agent that decreases the amount of activated CNS lymphocytes, which results in anti-inflammatory and antiproliferative effects.

Product Page

In Stock(5 business days)  
BRC0758
Product IDBRC0758
Product classBioreference compound
CAS number53716-49-7
MW273.7
Synonyms
C 5720, Carprodyl, Imadyl, NSC 297935, Rimadyl, Ro 20-5720, Ro 20-5720/000
Transport conditionsNormal

Carprofen

Carprofen is a non-steroidal anti-inflammatory drug that selectively inhibits cyclooxygenase-2 (COX-2). It is no longer used in the clinical setting, but is approved for use in dogs.

Product Page

In Stock(5 business days)  
BRC0479
Product IDBRC0479
Product classBioreference compound
CAS number530-78-9
MW281.2
Synonyms
Arlef, CI 440, CN 27544, INF 1837, NSC 219007, NSC 82699
Transport conditionsNormal

Flufenamic acid

Flufenamic acid is an anthranilic acid-derived nonsteroidal anti-inflammatory drug (NSAID) thought to exert its actions by a prostanoid-independent mechanism.

Product Page

In Stock(5 business days)  
BRC0980
Product IDBRC0980
Product classBioreference compound
CAS number4394-00-7
MW282.2
Synonyms
Lopac-N-0630; UP 83; NFA; Niflugel; Actol; Donalgin; Nifluril;
Transport conditionsNormal

Niflumic Acid

Niflumic acid is a nonsteroidal anti-inflammatory fenamate, is a Ca2+-activated Cl- channel blocker. It inhibits both phospholipase A2 as well as COX-2.

Product Page

In Stock(5 business days)  
BRC0756
Product IDBRC0756
Product classBioreference compound
CAS number41340-25-4
MW287.4
Synonyms
Lodine, NIH 9918, NSC 282126, AY 24236
Transport conditionsNormal
Restrictions Included in California Proposition 65 list  WARNING! This product contains a chemical known to the State of California to cause birth defects or other reproductive harm. For more information go to www.P65Warnings.ca.gov.

Etodolac

Etodolac is a non-steroidal anti-inflammatory drug that selectively inhibits cyclooxygenase-2 (COX-2). It is an anti-inflammatory agent with analgesic and antipyretic properties.

Product Page

In Stock(5 business days)  
BRC0644
Product IDBRC0644
Product classBioreference compound
CAS number64461-82-1
MW290.2
Synonyms
AB 021, AN 021, DS 103-282, Sirdalud, Ternelin, Tizan
Transport conditionsNormal

Tizanidine hydrochloride

Tizanidine hydrochloride is an agonist at a2-adrenergic receptor sites (IC50 = 48 nM) and presumably reduces spasticity by increasing presynaptic inhibition of motor neurons.

Product Page

In Stock(5 business days)  
BRC0426
Product IDBRC0426
Product classBioreference compound
CAS number21256-18-8
MW293.3
Synonyms
WY-21743, Daypro, NSC 310839, Alvo
Transport conditionsNormal

Oxaprozin

Oxaprozin is a nonsteroidal anti-inflammatory drug (NSAID) with analgesic and antipyretic properties.

Product Page

In Stock(5 business days)  
BRC0518
Product IDBRC0518
Product classBioreference compound
CAS number2444-46-4
MW293.4
Synonyms
8-Nordihydrocapsaicin, AH 23491X, NSC 172795, Pseudocapsaicin
Transport conditionsNormal

Nonivamide

Nonivamide is an capsaicinoid. Like capsaicin, it can deter mammals (but not birds or insects) from consuming plants or seeds. Nonivamide is a TRPV1 ion channel agonist. Mammalian TRPV1 is activated by heat and capsaicin, but the avian form is insensitive to capsaicin.

Product Page

In Stock(5 business days)  
BRC0989
Product IDBRC0989
Product classBioreference compound
CAS number15307-86-5
MW296.2
Synonyms
ISV-205;
Transport conditionsNormal

Diclofenac

Diclofenac is a nonsteroidal anti-inflammatory drug with analgesic and antipyretic properties. It inhibits both leukocyte migration and the enzyme cyclooxygenase (COX-1 and COX-2), leading to the peripheral inhibition of prostaglandin synthesis.

Product Page

In Stock(5 business days)  
BRC0359
Product IDBRC0359
Product classBioreference compound
CAS number50-33-9
MW308.4
Synonyms
Butazolidinel
Transport conditionsNormal

Phenylbutazone

Phenylbutazone is a compound of research interest as an anti-inflammatory and anti-proliferative agent.

Product Page

In Stock(5 business days)  
BRC0345
Product IDBRC0345
Product classBioreference compound
CAS number24237-54-5
MW316.4
Synonyms
Y-3642, Nonflamin, Dimaten
Transport conditionsNormal

Tinoridine

Tinoridine, also known as Y-3642, is a non-steroidal anti-inflammatory drug.

Product Page

In Stock(5 business days)  
BRC0166
Product IDBRC0166
Product classBioreference compound
CAS number67254-91-5
MW318.1
Synonyms
Meclofenamate, Arquel, Acide meclofenamique, Meclomen
Transport conditionsNormal

Meclofenamate sodium

A non-steroidal anti-inflammatory agent with antipyretic and antigranulation activities. It also inhibits prostaglandin biosynthesis.

Product Page

In Stock(5 business days)  
BRC0193
Product IDBRC0193
Product classBioreference compound
CAS number129-20-4
MW324.4
Synonyms
USAF Ge-14;
Transport conditionsNormal

Oxyphenbutazone

Oxyphenbutazone is a metabolite of Phenylbutazone. It is described to produce anti-inflammatory effects and demonstrates inhibition of cytokine production.

Product Page

In Stock(5 business days)  
BRC0232
Product IDBRC0232
Product classBioreference compound
CAS number130-95-0
MW324.4
Synonyms
(-)-Quinine, (8S,9R)-Quinine, Chinin, Jasoquin, QSM, Sulquin
Transport conditionsNormal

Quinine

Quinine is used parenterally to treat life-threatening infections caused by chloroquine-resistant Plasmodium falciparum malaria. Quinine acts as a blood schizonticide although it also has gametocytocidal activity against P. vivax and P. malariae.

Product Page

In Stock(5 business days)  
BRC0415
Product IDBRC0415
Product classBioreference compound
CAS number36322-90-4
MW331.4
Synonyms
Feldene; Larapam; NSC 666076; CP 16171; Bruxicam; Dolonex; Erazon; Improntal; Roxam; Roxiden; Sasulen; Solocalm; Trast;
Transport conditionsNormal

Piroxicam

Piroxicam is in a class of drugs called nonsteroidal anti-inflammatory drugs (NSAIDs). Piroxicam works by reducing hormones that cause inflammation and pain in the body.

Product Page

In Stock(5 business days)  
BRC0736
Product IDBRC0736
Product classBioreference compound
CAS number136434-34-9
MW333.9
Synonyms
LY 248686 HCl, Yentreve
Transport conditionsNormal

Duloxetine hydrochloride

Duloxetine is a potent inhibitor of neuronal serotonin and norepinephrine reuptake and a less potent inhibitor of dopamine reuptake. The antidepressant and pain inhibitory actions of duloxetine are believed to be related to its potentiation of serotonergic and noradrenergic activity in the CNS.

Product Page

In Stock(5 business days)  
BRC0810
Product IDBRC0810
Product classBioreference compound
CAS number581809-67-8
MW345.3
Synonyms
Transport conditionsNormal

A-425619

A-425619 is potent TRPV1 antagonist (IC50 = 3-9 nM). It blocks capsaicin-evoked currents in rat DRG neurons and inhibits TRPV1-activation by anandamide and N-arachidonoyl-dopamine. Reduces pain in inflammatory, postoperative and osteoarthritic in vivo pain models.

Product Page

In Stock(5 business days)  
BRC0797
Product IDBRC0797
Product classBioreference compound
CAS number71125-38-7
MW351.4
Synonyms
N1539, UH-AC 62XX
Transport conditionsNormal

Meloxicam

Meloxicam is an nonsteroidal anti-inflammatory drug with analgesic and antipyretic properties. It inhibits prostaglandin synthetase (cylooxygenase 1 and 2) and leads to a decrease of the synthesis of prostaglandins, therefore, inflammation is reduced.

Product Page

In Stock(5 business days)  
BRC0574
Product IDBRC0574
Product classBioreference compound
CAS number848057-98-7
MW354.3
Synonyms
MVRL1
Transport conditionsNormal

SPHINX

SPHINX is SRPK1 kinase inhibitor (IC50 = 440 nM).

Product Page

In Stock(5 business days)  
BRC0842
Product IDBRC0842
Product classBioreference compound
CAS number80573-04-2
MW357.3
Synonyms
Colazide, Giazo
Transport conditionsNormal

Balsalazide

Balsalazide is a prodrug that produce mesalamine (5-aminosalicylic acid), an anti inflammatory drug.

Product Page

In Stock(5 business days)  
BRC0367
Product IDBRC0367
Product classBioreference compound
CAS number53-86-1
MW357.8
Synonyms
Indocin
Transport conditionsNormal

Indomethacin

Indomethacin, an antiinflammatory agent, inhibits Cox-1 and Cox-2 (cyclooxygenases) with selectivity for Cox-1 (IC50 of 230 nM) over Cox-2 (IC50 of 630 nM). Additionally, indomethacin displays adipogenic actions via binding and activation of PPARγ (peroxisome proliferator-activated receptor γ), a ligand-activated transcription factor known to play an important role in adipogenesis.

Product Page

In Stock(5 business days)  
BRC0542
Product IDBRC0542
Product classBioreference compound
CAS number138926-19-9
MW359.2
Synonyms
BPH 24,
Transport conditionsNormal

Ibandronate sodium monohydrate

Ibandronate is a nitrogen-containing bisphosphonate, it binds to hydroxyapatite crystals with an affinity constant of 2.36 µM, inhibiting their growth and bone resorption.

Product Page

In Stock(5 business days)  
12
Display records per page

 

x
x