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CP21R7

Technical Data

Chemical name:CP21R7
Formula:C19H15N3O2
Molecular weight:317.3
CAS number:125314-13-8
SMILES:Cn1cc(C2=C(C(=O)NC2=O)c2cccc(N)c2)c2ccccc12 |t:4|

Cat. No. BRC0667

BRC0667

Prices

1.0 mg $ 112.0
2.0 mg $ 117.0
5.0 mg $ 126.0
10.0 mg $ 140.0
20.0 mg $ 250.0
25.0 mg $ 350.0

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Biological activity

It belongs to next groups of Bioreference compounds:
Target:

Kinases    Other kinases    Kinases    Enzyme-Linked Receptors    Receptor protein serine/threonine kinases   

Description:

CP21R7 is a potent and selective inhibitor of GSK3 beta (IC50 = 1.8 nM).

Targets:Glycogen synthase kinase-3 beta, Protein kinase C alpha type
References:
1. Bioorg. Med. Chem Letters. 2010; 20(5), 1693-1696.; 
2. PCT Int. Appl. 2012; WO 2012168167 A1 20121213.; 
3. PCT Int. Appl. 2017; WO 2017026878 A1 20170216.;