EnamineStore

Welcome, Guest
Tutorials

Return to Search menu

Debrisoquin

Isocaramidine, Bonipress, Declinax, Tendor

Technical Data

Chemical name:Debrisoquin
Formula:C10H14IN3
Molecular weight:303.1
CAS number:1052540-65-4
SMILES:I.NC(=N)N1CCc2ccccc2C1

Cat. No. BRC0357

BRC0357

Prices

1.0 mg $ 82.0
2.0 mg $ 84.0
5.0 mg $ 89.0
10.0 mg $ 116.0
20.0 mg $ 139.0
25.0 mg $ 151.0

Make inquiry

Biological activity

It belongs to next groups of Bioreference compounds:
Therapeutic areas:

Antihypertensive    Cardiovascular    CNS Agents    Neurotransmitter Agents   

Target:

Transporters    Ion Pumps    Neurotransmitter transporter   

Description:

Debrisoquin is an adrenergic neuron-blocking drug similar in effects to guanethidine. It is a substrate for a polymorphic cytochrome P-450 enzyme.

Targets:Sodium-dependent noradrenaline transporter
References:
1. Biochem. Pharmacol. 1969; 18: 891-901.; 
2. DNA. 1987; 6: 149-161.; 
3. Trends Pharmacol. 1989; Sci. 10: 107-109.; 
4. J. Chromatogr. B Biomed. Sci. Appl. 2000; 749: 153-161.;