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Chloroprocaine

Halestyn; Piocaine;

Technical Data

Chemical name:Chloroprocaine
Formula:C13H19ClN2O2
Molecular weight:270.8
CAS number:133-16-4
SMILES:CCN(CC)CCOC(=O)C1=C(Cl)C=C(N)C=C1

Cat. No. BRC0817

BRC0817

Prices

1.0 mg $ 83.0
2.0 mg $ 86.0
5.0 mg $ 91.0
10.0 mg $ 119.0
20.0 mg $ 205.0
25.0 mg $ 225.0

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Biological activity

It belongs to next groups of Bioreference compounds:
Therapeutic areas:

CNS Agents   

Target:

G-Protein-Coupled Receptors (GPCRs)    Dopamine receptor    5-hydroxytryptamine receptor (5-HT receptor) inhibitors    Glutamate receptor    Enzyme-Linked Receptors    Receptor protein serine/threonine kinases    Ion Channels    Sodium channel    Ligand-gated ion channels    Transporters    Ion Pumps    Neurotransmitter transporter   

Description:

Chloroprocaine is an anesthetic agent indicated for production of local or regional anesthesia. It blocks the generation and the conduction of nerve impulses, presumably by increasing the threshold for electrical excitation in the nerve, by slowing the propagation of the nerve impulse and by reducing the rate of rising of the action potential.

Targets:Sodium channel protein type 10 subunit alpha; Glutamate receptor ionotropic, NMDA 3A; Neuronal acetylcholine receptor subunit alpha-10; 5-hydroxytryptamine receptor 3A; Sodium-dependent dopamine transporter; Protein kinase C delta type;
References:
1. Eur J Pharmacol. 1995; 277, 1, 7 - 13.; 2. J Pharmacol Exp Ther. 2003; 306, 1, 84 - 92.; 3. US6391888, 2002, B1.;