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[3H]-YM 298198 Hydrochloride

Technical Data

Chemical name:[3H]-YM 298198 Hydrochloride
Formula:C18H23ClN4OS
Molecular weight:378.9
CAS number:1216398-09-2
SMILES:Cl.CN(C1CCCCC1)C(=O)C1=C(C)N2C(S1)=NC1=C2C=C(N)C=C1

Cat. No. BRC1085

BRC1085

Prices

1.0 mg $ 112.0
2.0 mg $ 117.0
5.0 mg $ 126.0
10.0 mg $ 140.0
20.0 mg $ 250.0
25.0 mg $ 350.0

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Biological activity

It belongs to next groups of Bioreference compounds:
Target:

G-Protein-Coupled Receptors (GPCRs)    Glutamate receptor   

Description:

YM 298198 hydrochloride is noncompetitive antagonist selective for mGluR-1. This compound also displays the ability to inhibit glutamate-induced IP production more potently than CPCCOEt.

Targets:Metabotropic glutamate receptor 1; Calcitonin gene-related peptide receptors;
References:
1. Current Drug Targets. 2007; 8, 5, 651 - 681.; 2. J Pharmacol Exp Ther. 2007; 321, 3, 1144 - 1153.; 3. J Pharmacol Exp Ther. 2005; 315, 1, 163 - 169.;