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3-methyloxetan-3-yl 4-[3-(2-methoxypyridin-3-yl)pyrazolo[1,5-a]pyrimidin-5-yl]piperazine-1-carboxylate

Technical Data

Chemical name:3-methyloxetan-3-yl 4-[3-(2-methoxypyridin-3-yl)pyrazolo[1,5-a]pyrimidin-5-yl]piperazine-1-carboxylate
Formula:C21H24N6O4
Molecular weight:424.5
CAS number:1809862-74-5
SMILES:COC1=C(C=CC=N1)C1=C2N=C(C=CN2N=C1)N1CCN(CC1)C(=O)OC1(C)COC1

Cat. No. BRC0577

BRC0577

Prices

1.0 mg $ 253.0
2.0 mg $ 258.0
5.0 mg $ 273.0
10.0 mg $ 547.0
20.0 mg $ 820.0
25.0 mg $ 984.0

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Biological activity

It belongs to next groups of Bioreference compounds:
Therapeutic areas:

Analgesics    CNS Agents    Antipsychotics    Antiparkinson   

Target:

Kinases    Other kinases    Kinases   

Description:

The compound is potent, brain penetrant inhibitor of AP2-associated protein kinase 1 (IC50 = 4.7 nM).

Targets:AP2-associated protein kinase 1;
References:
1. PCT Int. Appl. 2015; WO 2015142714 A1 20150924.;