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Letrozole

CGS 20267, Femara

Technical Data

Chemical name:Letrozole
Formula:C17H11N5
Molecular weight:285.3
CAS number:112809-51-5
SMILES:N#Cc1ccc(cc1)C(c1ccc(cc1)C#N)n1cncn1

Cat. No. BRC0787

BRC0787

Prices

1.0 mg $ 86.0
2.0 mg $ 88.0
5.0 mg $ 94.0
10.0 mg $ 121.0
20.0 mg $ 146.0
25.0 mg $ 159.0

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Biological activity

It belongs to next groups of Bioreference compounds:
Therapeutic areas:

Anti-cancer agents    Steroids   

Target:

Enzymes    Cytochrome P450 (CYP)    Aromatases   

Description:

Letrozole is an aromatase inhibitor used in the treatment of breast cancer.

Targets:Cytochrome P450 19A1 (aromatase)
References:
1. Bioorg. Med. Chem. 2012; 20, 7, 2427.; 
2. J. Med. Chem. 2012; 55, 19, 8464.; 
3. Cancer Res. 2006; 66, 23, 11485.;