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Enalaprilat dihydrate

Enalapril acid, MK-422 Dihydrate

Technical Data

Chemical name:Enalaprilat dihydrate
Formula:C18H28N2O7
Molecular weight:384.4
CAS number:84680-54-6
SMILES:O.O.C[C@H](N[C@@H](CCc1ccccc1)C(O)=O)C(=O)N1CCC[C@H]1C(O)=O

Cat. No. BRC0095

BRC0095

Prices

1.0 mg $ 55.0
2.0 mg $ 56.0
5.0 mg $ 59.0
10.0 mg $ 78.0
20.0 mg $ 93.0
25.0 mg $ 100.0

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Biological activity

It belongs to next groups of Bioreference compounds:
Therapeutic areas:

Antihypertensive   

Target:

G-Protein-Coupled Receptors (GPCRs)    Angiotensin receptor    Proteases    Proteases    Angiotensin-converting enzyme (ACE)    Renin angiotensin aldosterone system (RAAS) inhibitors   

Description:

Enalaprilat is the active metabolite of the orally available pro-drug, enalapril. Used in the treatment of hypertension, enalapril is an ACE inhibitor that prevents Angiotensin Converting Enzyme (ACE) from transforming angiotensin I into angiotensin II.

Targets:Angiotensin-converting enzyme
References:
1. Drug Metab Rev. 1983; 14(1):99-110.; 
2. Br J Clin Pharmacol. 1984; 18 Suppl 2:215S-229S.;