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Zoxazolamine

Flexin; McN-485; NSC 24995; Zoxamin;

Technical Data

Chemical name:Zoxazolamine
Formula:C7H5ClN2O
Molecular weight:168.6
CAS number:61-80-3
SMILES:NC1=NC2=C(O1)C=CC(Cl)=C2

Cat. No. BRC1044

BRC1044

Prices

1.0 mg $ 55.0
2.0 mg $ 56.0
5.0 mg $ 59.0
10.0 mg $ 78.0
20.0 mg $ 93.0
25.0 mg $ 100.0

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Biological activity

It belongs to next groups of Bioreference compounds:
Therapeutic areas:

Muscle relaxant   

Target:

Kinases    Mitogen-activated protein kinase (MAPK)    Kinases    Enzyme-Linked Receptors    Receptor protein serine/threonine kinases    Ion Channels    Potassium channel   

Description:

Zoxazolamine is a potent skeletal muscle relaxant that also has uricosuric activity. It is used as a tool for assessing hepatic cytochrome P-450 activity.

Targets:Calcium-activated potassium channel Small conductance (KCa2.1); Intermediate conductance calcium-activated potassium channel protein 4; 3-phosphoinositide-dependent protein kinase 1; Mitogen-activated protein kinase 1;
References:
1. Curr Med Chem. 2007; 14, 13, 1437 - 1457.; 2. The J Pharmacol Exp Ther. 2001; 296, 3, 683 - 689.; 3. Bioorg Med Chem Lett. 2015; 25, 21, 4728 - 4732.;